[Lys8]-Vasopressin TFA

Modify Date: 2024-01-02 19:15:12

[Lys8]-Vasopressin TFA structure	Common Name	[Lys8]-Vasopressin TFA
	CAS Number	50-57-7	Molecular Weight	1056.218
	Density	1.3±0.1 g/cm3	Boiling Point	1610.4±65.0 °C at 760 mmHg
	Molecular Formula	C₄₆H₆₅N₁₃O₁₂S₂	Melting Point	N/A
	MSDS	Chinese USA	Flash Point	927.7±34.3 °C
	Symbol	GHS07	Signal Word	Warning

Use of [Lys8]-Vasopressin TFA

Lysipressin is Antidiuretic hormone that have been found in pigs and some marsupial families. Induces contraction of the rabbit urinary bladder smooth muscle, activate adenylate-cyclase. Sequence: Cys-Tyr-Phe-Gln-Asn-Cys-Pro-Lys-Gly-NH2(Disulfide bridge: Cys1-Cys6).

Name	Lypressin
Synonym	More Synonyms

Description	Lysipressin is Antidiuretic hormone that have been found in pigs and some marsupial families. Induces contraction of the rabbit urinary bladder smooth muscle, activate adenylate-cyclase. Sequence: Cys-Tyr-Phe-Gln-Asn-Cys-Pro-Lys-Gly-NH2(Disulfide bridge: Cys1-Cys6).
Related Catalog	Signaling Pathways >> Others >> Others Research Areas >> Others Peptides
References	[1]. Gorbulev V et al. Molecular cloning and functional characterization of V2 [8-lysine] vasopressin and oxytocin receptors from a pig kidney cell line. Eur J Biochem. 1993 Jul 1;215(1):1-7. [2]. Crankshaw D et al. [Arg8]vasopressin-induced contractions of rabbit urinary bladder smooth muscle.Eur J Pharmacol. 1989 Dec 7;173(2-3):183-8.

Description

Related Catalog

Signaling Pathways >> Others >> Others

Research Areas >> Others

Peptides

References

[1]. Gorbulev V et al. Molecular cloning and functional characterization of V2 [8-lysine] vasopressin and oxytocin receptors from a pig kidney cell line. Eur J Biochem. 1993 Jul 1;215(1):1-7.

[2]. Crankshaw D et al. [Arg8]vasopressin-induced contractions of rabbit urinary bladder smooth muscle.Eur J Pharmacol. 1989 Dec 7;173(2-3):183-8.

Density	1.3±0.1 g/cm3
Boiling Point	1610.4±65.0 °C at 760 mmHg
Molecular Formula	C₄₆H₆₅N₁₃O₁₂S₂
Molecular Weight	1056.218
Flash Point	927.7±34.3 °C
Exact Mass	1055.431763
PSA	476.15000
LogP	-5.74
Vapour Pressure	0.0±0.3 mmHg at 25°C
Index of Refraction	1.581
Storage condition	−20°C

CHEMICAL IDENTIFICATION

RTECS NUMBER :: YW8659000

CHEMICAL NAME :: Vasopressin, 8-L-lysine-

CAS REGISTRY NUMBER :: 50-57-7

LAST UPDATED :: 199612

DATA ITEMS CITED :: 2

MOLECULAR FORMULA :: C46-H65-N13-O12-S2

MOLECULAR WEIGHT :: 1056.36

HEALTH HAZARD DATA

ACUTE TOXICITY DATA

TYPE OF TEST :: TDLo - Lowest published toxic dose

ROUTE OF EXPOSURE :: Intravenous

DOSE :: 5 iu/kg

SEX/DURATION :: female 12 day(s) after conception

TOXIC EFFECTS :: Reproductive - Effects on Embryo or Fetus - maternal-fetal exchange

REFERENCE :: JRPFA4 Journal of Reproduction and Fertility. (Biochemical Soc. Book Depot, POB 32, Commerce Way, Colchester, Essex CO2 8HP, UK) V.1- 1960- Volume(issue)/page/year: 17,419,1968

TYPE OF TEST :: TDLo - Lowest published toxic dose

ROUTE OF EXPOSURE :: Intraarterial

DOSE :: 0.25 iu/kg

SEX/DURATION :: female 12 day(s) after conception

TOXIC EFFECTS :: Reproductive - Effects on Embryo or Fetus - maternal-fetal exchange

REFERENCE :: JRPFA4 Journal of Reproduction and Fertility. (Biochemical Soc. Book Depot, POB 32, Commerce Way, Colchester, Essex CO2 8HP, UK) V.1- 1960- Volume(issue)/page/year: 17,419,1968

Symbol	GHS07
Signal Word	Warning
Hazard Statements	H332
Precautionary Statements	P261
Personal Protective Equipment	dust mask type N95 (US);Eyeshields;Gloves
Hazard Codes	Xn:Harmful;
Risk Phrases	R20
Safety Phrases	S36
RIDADR	NONH for all modes of transport
WGK Germany	3
RTECS	YW8659000

Precursor 0
DownStream 2
CAS#:63-91-2 L-Phenylalanine CAS#:60-18-4 L-Tyrosine

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EINECS 200-050-5

syntopressin

postacton

Lysipressin Acetate

CYFQNCPKG-NH2

LVP

[Lys8]-vasopressin

LYSPRESSIN

lypressin

8-lysine-vasopressin

lysinepitressin

diapid

lysine-vasopressin

Glycinamide, 1-[[(4R,7S,10S,13S,16S,19R)-19-amino-7-(2-amino-2-oxoethyl)-10-(3-amino-3-oxopropyl)-16-[(4-hydroxyphenyl)methyl]-6,9,12,15,18-pentaoxo-13-(phenylmethyl)-1,2-dithia-5,8,11,14,17-pentaazacycloeicos-4-yl]carbonyl]-L-prolyl-L-lysyl-

L-Cysteinyl-L-tyrosyl-L-phenylalanyl-L-glutaminyl-L-asparaginyl-L-cysteinyl-L-prolyl-L-lysylglycinamide Cyclic (1®6)-Disulfide

(8-Lysine)vasopressin

1-{[(4R,7S,10S,13S,16S,19R)-19-Amino-7-(2-amino-2-oxoethyl)-10-(3-amino-3-oxopropyl)-13-benzyl-16-(4-hydroxybenzyl)-6,9,12,15,18-pentaoxo-1,2-dithia-5,8,11,14,17-pentaazacycloicosan-4-yl]carbonyl}-L-prolyl-L-lysylglycinamide

Lysipressin

Lysine Vasopressin

Cys-Pro-Arg-Gly-NH2

c[Cys-Tyr-Phe-Gln-Asn-Cys]-Pro-Lys-Gly-NH2

CYS-TYR-PHE-GLN-ASN-CYS-PRO-LYS-GLY-NH2(DISULFIDE BRIDGE:CYS1-CYS6)

Lypressin Acetate