GPR4 antagonist 3
Modify Date: 2024-01-14 15:13:26
GPR4 antagonist 3 structure
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Common Name | GPR4 antagonist 3 | ||
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| CAS Number | 1401728-56-0 | Molecular Weight | 416.52 | |
| Density | N/A | Boiling Point | N/A | |
| Molecular Formula | C24H28N6O | Melting Point | N/A | |
| MSDS | N/A | Flash Point | N/A | |
Use of GPR4 antagonist 3GPR4 antagonist 3 is a selective, and orally available GPR4 antagonist with an IC50 of 70 nM[1]. Anti-inflammatory activities[1]. |
| Name | GPR4 antagonist 3 |
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| Description | GPR4 antagonist 3 is a selective, and orally available GPR4 antagonist with an IC50 of 70 nM[1]. Anti-inflammatory activities[1]. |
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| Related Catalog | |
| Target |
IC50: 70 nM (GPR4)[1]. |
| In Vivo | GPR4 antagonist 3 shows a significant anti-inflammatory effect in the rat antigen induced arthritis model after oral administration at 30 mg/kg bid[1].GPR4 antagonist 3 also prevents angiogenesis in the mouse chamber model as well as pain as demonstrated in the rat complete Freund’s adjuvant model[1]. |
| References |
| Molecular Formula | C24H28N6O |
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| Molecular Weight | 416.52 |