CRTh2 antagonist 3
Modify Date: 2024-01-13 10:45:08
CRTh2 antagonist 3 structure
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Common Name | CRTh2 antagonist 3 | ||
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| CAS Number | 312928-72-6 | Molecular Weight | 356.44 | |
| Density | N/A | Boiling Point | N/A | |
| Molecular Formula | C19H20N2O3S | Melting Point | N/A | |
| MSDS | N/A | Flash Point | N/A | |
Use of CRTh2 antagonist 3CRTh2 antagonist 3 is a potent chemoattractant receptor-homologous molecule expressed on Th2 cells (CRTh2) antagonist[1]. CRTh2 antagonist 3 (compound 4) also enhances the activity of PDK1 toward a short peptide substrate, with an EC50 of 2 μM and a Kd of 8.4 μM. CRTh2 antagonist 3 has the potential for cardiovascular inflammation[2]. |
| Name | CRTh2 antagonist 3 |
|---|
| Description | CRTh2 antagonist 3 is a potent chemoattractant receptor-homologous molecule expressed on Th2 cells (CRTh2) antagonist[1]. CRTh2 antagonist 3 (compound 4) also enhances the activity of PDK1 toward a short peptide substrate, with an EC50 of 2 μM and a Kd of 8.4 μM. CRTh2 antagonist 3 has the potential for cardiovascular inflammation[2]. |
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| Related Catalog | |
| Target |
CRTh2[1] EC50: 2 μM (PDK1)[2] Ki: 8.4 μM (PDK1)[2] |
| References |
| Molecular Formula | C19H20N2O3S |
|---|---|
| Molecular Weight | 356.44 |