Chemsrc provides Others's classification, including all related biologically active compounds cover the research fields of cancer, neuroscience, immunology and other popular diseases, etc.


Anti-infection >
Arenavirus Bacterial CMV Enterovirus Filovirus Fungal HBV HCV HIV HSV Influenza Virus Parasite Reverse Transcriptase RSV SARS-CoV
Antibody-drug Conjugate >
ADC Cytotoxin ADC Linker Drug-Linker Conjugates for ADC PROTAC-linker Conjugate for PAC
Apoptosis >
Apoptosis Bcl-2 Family c-Myc Caspase DAPK Ferroptosis IAP MDM-2/p53 PKD RIP kinase Survivin Thymidylate Synthase TNF Receptor
Autophagy >
Autophagy LRRK2 ULK Mitophagy
Cell Cycle/DNA Damage >
Antifolate APC ATM/ATR Aurora Kinase Casein Kinase CDK Checkpoint Kinase (Chk) CRISPR/Cas9 Deubiquitinase DNA Alkylator/Crosslinker DNA-PK DNA/RNA Synthesis Eukaryotic Initiation Factor (eIF) G-quadruplex Haspin Kinase HDAC HSP IRE1 Kinesin LIM Kinase (LIMK) Microtubule/Tubulin Mps1 Nucleoside Antimetabolite/Analog p97 PAK PARP PERK Polo-like Kinase (PLK) PPAR RAD51 ROCK Sirtuin SRPK Telomerase TOPK Topoisomerase Wee1
Cytoskeleton >
Arp2/3 Complex Dynamin Gap Junction Protein Integrin Kinesin Microtubule/Tubulin Mps1 Myosin PAK
Epigenetics >
AMPK Aurora Kinase DNA Methyltransferase Epigenetic Reader Domain HDAC Histone Acetyltransferase Histone Demethylase Histone Methyltransferase JAK MicroRNA PARP PKC Sirtuin Protein Arginine Deiminase
GPCR/G Protein >
5-HT Receptor Adenosine Receptor Adenylate Cyclase Adiponectin Receptor Adrenergic Receptor Angiotensin Receptor Bombesin Receptor Bradykinin Receptor Cannabinoid Receptor CaSR CCR CGRP Receptor Cholecystokinin Receptor CRFR CXCR Dopamine Receptor EBI2/GPR183 Endothelin Receptor GHSR Glucagon Receptor Glucocorticoid Receptor GNRH Receptor GPCR19 GPR109A GPR119 GPR120 GPR139 GPR40 GPR55 GPR84 Guanylate Cyclase Histamine Receptor Imidazoline Receptor Leukotriene Receptor LPL Receptor mAChR MCHR1 (GPR24) Melatonin Receptor mGluR Motilin Receptor Neurokinin Receptor Neuropeptide Y Receptor Neurotensin Receptor Opioid Receptor Orexin Receptor (OX Receptor) Oxytocin Receptor P2Y Receptor Prostaglandin Receptor Protease-Activated Receptor (PAR) Ras RGS Protein Sigma Receptor Somatostatin Receptor TSH Receptor Urotensin Receptor Vasopressin Receptor Melanocortin Receptor
Immunology/Inflammation >
Aryl Hydrocarbon Receptor CCR Complement System COX CXCR FLAP Histamine Receptor IFNAR Interleukin Related IRAK MyD88 NO Synthase NOD-like Receptor (NLR) PD-1/PD-L1 PGE synthase Salt-inducible Kinase (SIK) SPHK STING Thrombopoietin Receptor Toll-like Receptor (TLR) Arginase
JAK/STAT Signaling >
EGFR JAK Pim STAT
MAPK/ERK Pathway >
ERK JNK KLF MAP3K MAP4K MAPKAPK2 (MK2) MEK Mixed Lineage Kinase MNK p38 MAPK Raf Ribosomal S6 Kinase (RSK)
Membrane Transporter/Ion Channel >
ATP Synthase BCRP Calcium Channel CFTR Chloride Channel CRAC Channel CRM1 EAAT2 GABA Receptor GlyT HCN Channel iGluR Monoamine Transporter Monocarboxylate Transporter Na+/Ca2+ Exchanger Na+/HCO3- Cotransporter Na+/K+ ATPase nAChR NKCC P-glycoprotein P2X Receptor Potassium Channel Proton Pump SGLT Sodium Channel TRP Channel URAT1
Metabolic Enzyme/Protease >
15-PGDH 5 alpha Reductase 5-Lipoxygenase Acetyl-CoA Carboxylase Acyltransferase Adenosine Deaminase Adenosine Kinase Aldehyde Dehydrogenase (ALDH) Aldose Reductase Aminopeptidase Angiotensin-converting Enzyme (ACE) ATGL ATP Citrate Lyase Carbonic Anhydrase Carboxypeptidase Cathepsin CETP COMT Cytochrome P450 Dipeptidyl Peptidase Dopamine β-hydroxylase E1/E2/E3 Enzyme Elastase Enolase FAAH FABP Factor Xa Farnesyl Transferase Fatty Acid Synthase (FAS) FXR Glucokinase GSNOR Gutathione S-transferase HCV Protease Hexokinase HIF/HIF Prolyl-Hydroxylase HIV Integrase HIV Protease HMG-CoA Reductase (HMGCR) HSP Indoleamine 2,3-Dioxygenase (IDO) Isocitrate Dehydrogenase (IDH) Lactate Dehydrogenase LXR MAGL Mineralocorticoid Receptor Mitochondrial Metabolism MMP Nampt NEDD8-activating Enzyme Neprilysin PAI-1 PDHK PGC-1α Phosphatase Phosphodiesterase (PDE) Phospholipase Procollagen C Proteinase Proteasome Pyruvate Kinase RAR/RXR Renin ROR Ser/Thr Protease SGK Stearoyl-CoA Desaturase (SCD) Thrombin Tryptophan Hydroxylase Tyrosinase Xanthine Oxidase
Neuronal Signaling >
5-HT Receptor AChE Adenosine Kinase Amyloid-β Beta-secretase CaMK CGRP Receptor COMT Dopamine Receptor Dopamine Transporter FAAH GABA Receptor GlyT iGluR Imidazoline Receptor mAChR Melatonin Receptor Monoamine Oxidase nAChR Neurokinin Receptor Opioid Receptor Serotonin Transporter γ-secretase
NF-κB >
NF-κB IKK Keap1-Nrf2 MALT1
PI3K/Akt/mTOR >
Akt AMPK ATM/ATR DNA-PK GSK-3 MELK mTOR PDK-1 PI3K PI4K PIKfyve PTEN
PROTAC >
PROTAC E3 Ligase Ligand-Linker Conjugate Ligand for E3 Ligase PROTAC Linker PROTAC-linker Conjugate for PAC
Protein Tyrosine Kinase/RTK >
Ack1 ALK Bcr-Abl BMX Kinase Btk c-Fms c-Kit c-Met/HGFR Discoidin Domain Receptor DYRK EGFR Ephrin Receptor FAK FGFR FLT3 IGF-1R Insulin Receptor IRAK Itk PDGFR PKA Pyk2 ROS Src Syk TAM Receptor Trk Receptor VEGFR
Stem Cell/Wnt >
Casein Kinase ERK Gli GSK-3 Hedgehog Hippo (MST) JAK Notch Oct3/4 PKA Porcupine ROCK sFRP-1 Smo STAT TGF-beta/Smad Wnt YAP β-catenin γ-secretase
TGF-beta/Smad >
TGF-beta/Smad PKC ROCK TGF-β Receptor
Vitamin D Related >
VD/VDR
Others >
Androgen Receptor Aromatase Estrogen Receptor/ERR Progesterone Receptor Thyroid Hormone Receptor Others

Methyl L-phenylalaninate hydrochloride

H-Phe-OMe.hydrochloride is a phenylalanine derivative[1].

  • CAS Number: 7524-50-7
  • MF: C10H14ClNO2
  • MW: 215.677
  • Catalog: Others
  • Density: N/A
  • Boiling Point: 264.2ºC at 760 mmHg
  • Melting Point: 156-160ºC
  • Flash Point: 126ºC

H-Arg-Ser-Arg-OH acetate salt

H-Arg-Ser-Arg-OH is a short peptide. H-Arg-Ser-Arg-OH is a motif of di-leucine and RSRR, it can be used to design larger peptides and compound[1].

  • CAS Number: 115035-42-2
  • MF: C15H31N9O5
  • MW: 417.46400
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

SPDP

SPDP is a short-chain crosslinker for amine-to-sulfhydryl conjugation via NHS-ester and pyridyldithiol reactive groups that form cleavable (reducible) disulfide bonds with cysteine sulfhydryls. equal amounts of anti-CD11c and anti-CTLA-4 Abs (in borate buffered saline; pH 8.5) were activated using SPDP .

  • CAS Number: 68181-17-9
  • MF: C12H12N2O4S2
  • MW: 312.365
  • Catalog: Others
  • Density: 1.5±0.1 g/cm3
  • Boiling Point: 465.9±55.0 °C at 760 mmHg
  • Melting Point: 84-86 °C(lit.)
  • Flash Point: 235.6±31.5 °C

N-Acetyl-D-lactosamine

N-Acetyllactosamine (LacNAc), a nitrogen-containing disaccharide, is an important component of various oligosaccharides such as glycoproteins and sialyl Lewis X. N-Acetyllactosamine can be used as the starting material for the synthesis of various oligosaccharides. N-Acetyllactosamine has prebiotic effects[1][2].

  • CAS Number: 32181-59-2
  • MF: C14H25NO11
  • MW: 383.34800
  • Catalog: Others
  • Density: 1.64 g/cm3
  • Boiling Point: 805.5ºC at 760 mmHg
  • Melting Point: 191-192ºC
  • Flash Point: 441ºC

D-Galactose-13C-1

D-Galactose-13C-1 is the 13C labeled D-galactopyranose[1].

  • CAS Number: 314062-47-0
  • MF: C6H12O6
  • MW: 181.14900
  • Catalog: Others
  • Density: 1.732g/cm3
  • Boiling Point: N/A
  • Melting Point: 170-172ºC(lit.)
  • Flash Point: N/A

Fmoc-N-methyl--D-phenylalanine

N-[(9H-Fluoren-9-ylmethoxy)carbonyl]-N-methyl-D-phenylalanine is a phenylalanine derivative[1].

  • CAS Number: 138775-05-0
  • MF: C25H23NO4
  • MW: 401.454
  • Catalog: Others
  • Density: 1.3±0.1 g/cm3
  • Boiling Point: 595.4±39.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 313.9±27.1 °C

Calpain-1 (pig)

Calpain-1 (pig) (μ-Calpain) is an intracellular Ca2+-regulated cysteine protease. Calpain-1 (pig) exhibits neuroprotective effect[1][2].

  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Fura-2, AM

Fura-2 AM is a ratiometric fluorescent Ca2+ indicator.

  • CAS Number: 108964-32-5
  • MF: C44H47N3O24
  • MW: 1001.850
  • Catalog: Dye Reagents
  • Density: 1.4±0.1 g/cm3
  • Boiling Point: 975.9±75.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 544.0±37.1 °C

GalNAc beta(1-4)GlcNAc-beta-pNP

GalNAcβ(1-4)GlcNAc-β-pNP is a biochemical reagent that can be used as a biological material or organic compound for life science related research.

  • CAS Number: 872578-72-8
  • MF: C22H31N3O13
  • MW: 545.49400
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

1,1,1,3,10,11-Hexachloroundecane

1,1,1,3,10,11-Hexachloroundecane is a kind of polychlorinated alkane (PCA) that has a long carbon chain length[1].

  • CAS Number: 601523-28-8
  • MF: C11H18Cl6
  • MW: 362.979
  • Catalog: Others
  • Density: 1.3±0.1 g/cm3
  • Boiling Point: 384.5±10.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 176.1±16.4 °C

ALANINE, N-[[4-(2-CHLOROPHENOXY)PHENYL]SULFONYL]

N-[4-(2-Chlorophenoxy)phenylsulfonyl]-DL-alanine is an alanine derivative[1].

  • CAS Number: 1008472-78-3
  • MF: C15H14ClNO5S
  • MW: 355.79300
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

5-Bromo(3,3,4,4-2H4)pentanoic acid

5-Bromopentanoic-3,3,4,4 Acid-d4 is the deuterium labeled 5-Bromopentanoic acid[1].

  • CAS Number: 42932-62-7
  • MF: C5H5BrD4O2
  • MW: 185.052
  • Catalog: Others
  • Density: 1.5±0.1 g/cm3
  • Boiling Point: 265.5±23.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 114.4±22.6 °C

Indole-3-acetamide-d5

Indole-3-acetamide-d5 is the deuterium labeled Indole-3-acetamide[1]. Indole-3-acetamide is a biosynthesis intermediate of indole-3-acetic acid (HY-18569). Indole-3-acetic acid is the most common natural plant growth hormone of the auxin class[2].

  • CAS Number: 1204700-53-7
  • MF: C10H10N2O
  • MW: 174.199
  • Catalog: Others
  • Density: 1.3±0.1 g/cm3
  • Boiling Point: 407.1±47.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 200.0±29.3 °C

1,8-Dichloroanthraquinone

1,8-Dichloroanthraquinone, an anthraquinone, is an inhibitor of sulfide production by sulfate-reducing bacteria[1].

  • CAS Number: 82-43-9
  • MF: C14H6Cl2O2
  • MW: 277.10
  • Catalog: Bacterial
  • Density: 1.5±0.1 g/cm3
  • Boiling Point: 455.2±45.0 °C at 760 mmHg
  • Melting Point: 201.5-203 °C(lit.)
  • Flash Point: 191.7±29.3 °C

Isovalerylcarnitine

Isovalerylcarnitine is a product of the catabolism of L-leucine. It increases calpain activity.

  • CAS Number: 31023-24-2
  • MF: C12H23NO4
  • MW: 245.31500
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Boc-L-Cyclopentylglycine

(S)-2-((tert-Butoxycarbonyl)amino)-2-cyclopentylacetic acid is a Glycine (HY-Y0966) derivative[1].

  • CAS Number: 109183-72-4
  • MF: C12H21NO4
  • MW: 243.299
  • Catalog: Others
  • Density: 1.1±0.1 g/cm3
  • Boiling Point: 363.2±21.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 173.5±22.1 °C

Methyl p-hydroxyphenyllactate

Methyl p-hydroxyphenyllactate (MeHPLA) is an important cell growth-regulating agent which binds to nuclear type II binding sites in normal and malignant cells[1].

  • CAS Number: 51095-47-7
  • MF: C10H12O4
  • MW: 196.20
  • Catalog: Others
  • Density: 1.3±0.1 g/cm3
  • Boiling Point: 356.2±27.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 141.8±17.2 °C

C15 Ceramide-1-phosphate-d7

C15 Ceramide-1-phosphate-d7 is deuterium labeled C15 Ceramide-1-phosphate.

  • CAS Number: 2315262-27-0
  • MF: C33H62D7N2O6P
  • MW: 627.93
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

LITHIUM 3,5-DIIODOSALICYLATE

Lithium 3,5-diiodosalicylate is a biochemical reagent that can be used as a biological material or organic compound for life science related research.

  • CAS Number: 653-14-5
  • MF: C7H3I2LiO3
  • MW: 395.84700
  • Catalog: Others
  • Density: N/A
  • Boiling Point: 380.8ºC at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 184.1ºC

Substance P (free acid)

Substance P, Free Acid is a native substance P analog, but shows no biological activity of substance P.

  • CAS Number: 71977-09-8
  • MF: C63H97N17O14S
  • MW: 1348.61000
  • Catalog: Peptides
  • Density: 1.41 g/cm3
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Prodan

Prodan, a solvatochromic fluorophore, has been used as a microenvironment-sensitive membrane reporter. Based on the chemistry of Prodan, fluorescent nucleosides are designed and synthesized.The fluorescent nucleosides sensitively varied the Stokes shift values depending on the orientational polarizability of the solvent[1].

  • CAS Number: 70504-01-7
  • MF: C15H17NO
  • MW: 227.30200
  • Catalog: Others
  • Density: 1.085g/cm3
  • Boiling Point: 386.157ºC at 760 mmHg
  • Melting Point: 137ºC(lit.)
  • Flash Point: 150.15ºC

Tributyl citrate

Tributyl citrate is a citric acid ester. Tributyl citrate can be used as an excipient, such as plasticizer. Pharmaceutical excipients, or pharmaceutical auxiliaries, refer to other chemical substances used in the pharmaceutical process other than pharmaceutical ingredients. Pharmaceutical excipients generally refer to inactive ingredients in pharmaceutical preparations, which can improve the stability, solubility and processability of pharmaceutical preparations. Pharmaceutical excipients also affect the absorption, distribution, metabolism, and elimination (ADME) processes of co-administered drugs[1][2].

  • CAS Number: 77-94-1
  • MF: C18H32O7
  • MW: 360.45
  • Catalog: Others
  • Density: 1.1±0.1 g/cm3
  • Boiling Point: 389.8±9.0 °C at 760 mmHg
  • Melting Point: ≥300 °C(lit.)
  • Flash Point: 120.7±12.2 °C

Nitazoxanide D4

Nitazoxanide D4 is the deuterium labeled Nitazoxanide, which is an antiprotozoal agent.

  • CAS Number: 1246819-17-9
  • MF: C12H5D4N3O5S
  • MW: 311.30700
  • Catalog: Influenza Virus
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Arnidiol

Arnidiol is a pentacyclic triterpene isolated from Barleria Longiflora Linn F.[1].

  • CAS Number: 6750-30-7
  • MF: C30H50O2
  • MW: 442.717
  • Catalog: Others
  • Density: 1.0±0.1 g/cm3
  • Boiling Point: 518.2±43.0 °C at 760 mmHg
  • Melting Point: 257℃
  • Flash Point: 208.8±22.8 °C

3,3',4,4'-Tetrachloro-1,1'-biphenyl-d6

3,3',4,4'-Tetrachloro-1,1'-biphenyl-d6 is the deuterium labeled 3,3',4,4'-Tetrachloro-1,1'-biphenyl[1].

  • CAS Number: 93952-23-9
  • MF: C12Cl4D6
  • MW: 298.02500
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

(R)-IDO/TDO-IN-1

(R)-IDO/TDO-IN-1 (compound 25) is an indoleamine-2,3-dioxygenase (IDO) inhibitor, with good pharmacokinetic properties. (R)-IDO/TDO-IN-1 exhibits anti-tumor activity in MC38 xenograft model. (R)-IDO/TDO-IN-1 shows synergistic effect with anti-PD-1 monoclonal antibody (SHR-1210)[1].

  • CAS Number: 2033173-00-9
  • MF: C25H24FN5
  • MW: 413.49
  • Catalog: Indoleamine 2,3-Dioxygenase (IDO)
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

RET-IN-12

RET-IN-12 (compound 2) is a RET inhibitor, with IC50 values of 0.3 nM and 1 nM for RET(WT) and RET(V804M), respectively[1].

  • CAS Number: 2684252-55-7
  • MF: C30H30F3N5O4
  • MW: 581.59
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

(BHQ-3)-OSu hexafluorophosphate

(BHQ-3)-OSu hexafluorophosphate is used for fluorescent labeling of protease substrates[1].

  • CAS Number: 871240-95-8
  • MF: C37H38F6N7O4P
  • MW: 789.71
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

GW806742X

GW806742X is a Mixed Lineage Kinase Domain-Like (MLKL) inhibitor which binds the MLKL pseudokinase domain with a Kd value of 9.3 μM and anti-necroptosis activity. GW806742X has activity against VEGFR2[1][2].

  • CAS Number: 579515-63-2
  • MF: C25H22F3N7O4S
  • MW: 573.55
  • Catalog: Mixed Lineage Kinase
  • Density: 1.5±0.1 g/cm3
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

8-Hydroxyquinoline

8-Hydroxyquinoline is a monoprotic bidentate chelating agent, exhibits antiseptic, disinfectant, and pesticide properties, functioning as a transcription inhibitor.

  • CAS Number: 148-24-3
  • MF: C9H7NO
  • MW: 145.158
  • Catalog: Others
  • Density: 1.3±0.1 g/cm3
  • Boiling Point: 267.0±0.0 °C at 760 mmHg
  • Melting Point: 70-73 °C(lit.)
  • Flash Point: 143.1±20.4 °C