Chemsrc provides Others's classification, including all related biologically active compounds cover the research fields of cancer, neuroscience, immunology and other popular diseases, etc.


Anti-infection >
Arenavirus Bacterial CMV Enterovirus Filovirus Fungal HBV HCV HIV HSV Influenza Virus Parasite Reverse Transcriptase RSV SARS-CoV
Antibody-drug Conjugate >
ADC Cytotoxin ADC Linker Drug-Linker Conjugates for ADC PROTAC-linker Conjugate for PAC
Apoptosis >
Apoptosis Bcl-2 Family c-Myc Caspase DAPK Ferroptosis IAP MDM-2/p53 PKD RIP kinase Survivin Thymidylate Synthase TNF Receptor
Autophagy >
Autophagy LRRK2 ULK Mitophagy
Cell Cycle/DNA Damage >
Antifolate APC ATM/ATR Aurora Kinase Casein Kinase CDK Checkpoint Kinase (Chk) CRISPR/Cas9 Deubiquitinase DNA Alkylator/Crosslinker DNA-PK DNA/RNA Synthesis Eukaryotic Initiation Factor (eIF) G-quadruplex Haspin Kinase HDAC HSP IRE1 Kinesin LIM Kinase (LIMK) Microtubule/Tubulin Mps1 Nucleoside Antimetabolite/Analog p97 PAK PARP PERK Polo-like Kinase (PLK) PPAR RAD51 ROCK Sirtuin SRPK Telomerase TOPK Topoisomerase Wee1
Cytoskeleton >
Arp2/3 Complex Dynamin Gap Junction Protein Integrin Kinesin Microtubule/Tubulin Mps1 Myosin PAK
Epigenetics >
AMPK Aurora Kinase DNA Methyltransferase Epigenetic Reader Domain HDAC Histone Acetyltransferase Histone Demethylase Histone Methyltransferase JAK MicroRNA PARP PKC Sirtuin Protein Arginine Deiminase
GPCR/G Protein >
5-HT Receptor Adenosine Receptor Adenylate Cyclase Adiponectin Receptor Adrenergic Receptor Angiotensin Receptor Bombesin Receptor Bradykinin Receptor Cannabinoid Receptor CaSR CCR CGRP Receptor Cholecystokinin Receptor CRFR CXCR Dopamine Receptor EBI2/GPR183 Endothelin Receptor GHSR Glucagon Receptor Glucocorticoid Receptor GNRH Receptor GPCR19 GPR109A GPR119 GPR120 GPR139 GPR40 GPR55 GPR84 Guanylate Cyclase Histamine Receptor Imidazoline Receptor Leukotriene Receptor LPL Receptor mAChR MCHR1 (GPR24) Melatonin Receptor mGluR Motilin Receptor Neurokinin Receptor Neuropeptide Y Receptor Neurotensin Receptor Opioid Receptor Orexin Receptor (OX Receptor) Oxytocin Receptor P2Y Receptor Prostaglandin Receptor Protease-Activated Receptor (PAR) Ras RGS Protein Sigma Receptor Somatostatin Receptor TSH Receptor Urotensin Receptor Vasopressin Receptor Melanocortin Receptor
Immunology/Inflammation >
Aryl Hydrocarbon Receptor CCR Complement System COX CXCR FLAP Histamine Receptor IFNAR Interleukin Related IRAK MyD88 NO Synthase NOD-like Receptor (NLR) PD-1/PD-L1 PGE synthase Salt-inducible Kinase (SIK) SPHK STING Thrombopoietin Receptor Toll-like Receptor (TLR) Arginase
JAK/STAT Signaling >
EGFR JAK Pim STAT
MAPK/ERK Pathway >
ERK JNK KLF MAP3K MAP4K MAPKAPK2 (MK2) MEK Mixed Lineage Kinase MNK p38 MAPK Raf Ribosomal S6 Kinase (RSK)
Membrane Transporter/Ion Channel >
ATP Synthase BCRP Calcium Channel CFTR Chloride Channel CRAC Channel CRM1 EAAT2 GABA Receptor GlyT HCN Channel iGluR Monoamine Transporter Monocarboxylate Transporter Na+/Ca2+ Exchanger Na+/HCO3- Cotransporter Na+/K+ ATPase nAChR NKCC P-glycoprotein P2X Receptor Potassium Channel Proton Pump SGLT Sodium Channel TRP Channel URAT1
Metabolic Enzyme/Protease >
15-PGDH 5 alpha Reductase 5-Lipoxygenase Acetyl-CoA Carboxylase Acyltransferase Adenosine Deaminase Adenosine Kinase Aldehyde Dehydrogenase (ALDH) Aldose Reductase Aminopeptidase Angiotensin-converting Enzyme (ACE) ATGL ATP Citrate Lyase Carbonic Anhydrase Carboxypeptidase Cathepsin CETP COMT Cytochrome P450 Dipeptidyl Peptidase Dopamine β-hydroxylase E1/E2/E3 Enzyme Elastase Enolase FAAH FABP Factor Xa Farnesyl Transferase Fatty Acid Synthase (FAS) FXR Glucokinase GSNOR Gutathione S-transferase HCV Protease Hexokinase HIF/HIF Prolyl-Hydroxylase HIV Integrase HIV Protease HMG-CoA Reductase (HMGCR) HSP Indoleamine 2,3-Dioxygenase (IDO) Isocitrate Dehydrogenase (IDH) Lactate Dehydrogenase LXR MAGL Mineralocorticoid Receptor Mitochondrial Metabolism MMP Nampt NEDD8-activating Enzyme Neprilysin PAI-1 PDHK PGC-1α Phosphatase Phosphodiesterase (PDE) Phospholipase Procollagen C Proteinase Proteasome Pyruvate Kinase RAR/RXR Renin ROR Ser/Thr Protease SGK Stearoyl-CoA Desaturase (SCD) Thrombin Tryptophan Hydroxylase Tyrosinase Xanthine Oxidase
Neuronal Signaling >
5-HT Receptor AChE Adenosine Kinase Amyloid-β Beta-secretase CaMK CGRP Receptor COMT Dopamine Receptor Dopamine Transporter FAAH GABA Receptor GlyT iGluR Imidazoline Receptor mAChR Melatonin Receptor Monoamine Oxidase nAChR Neurokinin Receptor Opioid Receptor Serotonin Transporter γ-secretase
NF-κB >
NF-κB IKK Keap1-Nrf2 MALT1
PI3K/Akt/mTOR >
Akt AMPK ATM/ATR DNA-PK GSK-3 MELK mTOR PDK-1 PI3K PI4K PIKfyve PTEN
PROTAC >
PROTAC E3 Ligase Ligand-Linker Conjugate Ligand for E3 Ligase PROTAC Linker PROTAC-linker Conjugate for PAC
Protein Tyrosine Kinase/RTK >
Ack1 ALK Bcr-Abl BMX Kinase Btk c-Fms c-Kit c-Met/HGFR Discoidin Domain Receptor DYRK EGFR Ephrin Receptor FAK FGFR FLT3 IGF-1R Insulin Receptor IRAK Itk PDGFR PKA Pyk2 ROS Src Syk TAM Receptor Trk Receptor VEGFR
Stem Cell/Wnt >
Casein Kinase ERK Gli GSK-3 Hedgehog Hippo (MST) JAK Notch Oct3/4 PKA Porcupine ROCK sFRP-1 Smo STAT TGF-beta/Smad Wnt YAP β-catenin γ-secretase
TGF-beta/Smad >
TGF-beta/Smad PKC ROCK TGF-β Receptor
Vitamin D Related >
VD/VDR
Others >
Androgen Receptor Aromatase Estrogen Receptor/ERR Progesterone Receptor Thyroid Hormone Receptor Others

Protoapigenin

Protoapigenin is a flavonoid, that can be isolated from the aerial parts of Macrothelypteris torresiana[1].

  • CAS Number: 879325-07-2
  • MF: C15H12O6
  • MW: 288.25
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Z-Val-Lys-Met-AMC acetate salt

Z-Val-Lys-Met-AMC is a fluorescent substrate that can be used to detect the β-secretase activity of cathepsin B[1].

  • CAS Number: 141223-71-4
  • MF: C34H45N5O7S
  • MW: 667.82
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

N,N-Bis(carboxymethyl)-L-lysine

Nα,Nα-Bis(carboxymethyl)-L-lysine is a competitive inhibitor of bitter taste receptor 4, with an IC50 of 59 nM. Nα,Nα-Bis(carboxymethyl)-L-lysine can be used in bitter receptors related study[1][2][3].

  • CAS Number: 113231-05-3
  • MF: C10H18N2O6
  • MW: 262.26
  • Catalog: Others
  • Density: 1.4±0.1 g/cm3
  • Boiling Point: 537.8±50.0 °C at 760 mmHg
  • Melting Point: >208°C
  • Flash Point: 279.0±30.1 °C

3β,5α,6β-Trihydroxycholestane

3β,5α,6β-Trihydroxycholestane is a biochemical reagent that can be used as a biological material or organic compound for life science related research.

  • CAS Number: 1253-84-5
  • MF: C27H48O3
  • MW: 420.668
  • Catalog: Others
  • Density: 1.1±0.1 g/cm3
  • Boiling Point: 515.7±40.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 212.5±21.9 °C

Methyl isovanillate

Methyl isovanillate is a secondary metabolite isolated from Vitex agnus-castus[1].

  • CAS Number: 6702-50-7
  • MF: C9H10O4
  • MW: 182.173
  • Catalog: Others
  • Density: 1.2±0.1 g/cm3
  • Boiling Point: 327.7±22.0 °C at 760 mmHg
  • Melting Point: 64-67ºC
  • Flash Point: 132.8±15.8 °C

Pseudoaspidin

Pseudoaspidin is isolated from the ferns of the class Pterophyta or Filicinae[1].

  • CAS Number: 478-28-4
  • MF: C25H32O8
  • MW: 460.51700
  • Catalog: Others
  • Density: N/A
  • Boiling Point: 647.7±55.0 °C
  • Melting Point: 142-144 °C
  • Flash Point: N/A

Hoechst 33258 analog 3

Hoechst stains are part of a family of blue fluorescent dyes used to stain DNA.IC50 Value:Target: These Bis-benzimides were originally developed by Hoechst AG, which numbered all their compounds so that the dye Hoechst 33342 is the 33342nd compound made by the company. There are three related Hoechst stains: Hoechst 33258, Hoechst 33342, and Hoechst 34580. The dyes Hoechst 33258 and Hoechst 33342 are the ones most commonly used and they have similarexcitation/emission spectra. Both dyes are excited by ultraviolet light at around 350 nm, and both emit blue/cyan fluorescent light around anemission maximum at 461 nm. Unbound dye has its maximum fluorescence emission in the 510-540 nm range. Hoechst dyes are soluble in water and in organic solvents such as dimethyl formamide or dimethyl sulfoxide. Concentrations can be achieved of up to 10 mg/mL. Aqueous solutions are stable at 2-6 °C for at least six months when protected from light. For long-term storage the solutions are instead frozen at ≤-20 °C.The dyes bind to the minor groove of double-stranded DNA with a preference for sequences rich in adenine andthymine. Although the dyes can bind to all nucleic acids, AT-rich double-stranded DNA strands enhance fluorescence considerably.Hoechst dyes are cell-permeable and can bind to DNA in live or fixed cells. Therefore, these stains are often called supravital, which means that cells survive a treatment with these compounds. Cells that express specific ATP-binding cassette transporter proteins can also actively transport these stains out of their cytoplasm.

  • CAS Number: 23554-98-5
  • MF: C26H26N6
  • MW: 422.52500
  • Catalog: Dye Reagents
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Fmoc-Asn(Dmcp)-OH

Fmoc-Asn(Dmcp)-OH is an asparagine derivative[1].

  • CAS Number: 172947-19-2
  • MF: C25H28N2O5
  • MW: 436.50000
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

D-Alanine ethyl ester hydrochloride

D-Alanine ethyl ester hydrochloride is an alanine derivative[1].

  • CAS Number: 6331-09-5
  • MF: C5H12ClNO2
  • MW: 153.607
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Acetyl Hexapeptide-1

Acetyl hexapeptide-1 (Melitane) is a bioactive peptide with anti-wrinkle effect and has been reported used as a cosmetic ingredient[1].

  • CAS Number: 448944-47-6
  • MF: C43H59N13O7
  • MW: 870.011
  • Catalog: Others
  • Density: 1.4±0.1 g/cm3
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

D-Leucinol

D-Leucinol is the inactive isomer of L-Leucinol (HY-W015876), and can be used as an experimental control. L-Leucinol ((+)-Leucinol) is a competitive aminopeptidase inhibitor with Ki value of 17 μM[1].

  • CAS Number: 53448-09-2
  • MF: C6H15NO
  • MW: 117.19
  • Catalog: Others
  • Density: 0.9±0.1 g/cm3
  • Boiling Point: 198.6±0.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 78.6±19.8 °C

Levatin

Levatin is an 18-Norclerodane diterpene from Croton levatii[1].

  • CAS Number: 140670-84-4
  • MF: C19H20O5
  • MW: 328.35900
  • Catalog: Others
  • Density: 1.33g/cm3
  • Boiling Point: 578.4ºC at 760mmHg
  • Melting Point: N/A
  • Flash Point: 303.6ºC

Tenuifoliside C

Tenuifoliside C, isolated from polygala tenuifolia willd, significantly inhibits chlorzoxazone 6-hydroxylation catalyzed by CYP2E1[1].

  • CAS Number: 139726-37-7
  • MF: C35H44O19
  • MW: 768.71200
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Tricarballylic acid

Tricarballylic acid, a conjugate acid of a tricarballylate, is a competitive inhibitor of the enzyme aconitate hydratase (aconitase; EC 4.2.1.3) with a Ki value of 0.52 mM[1].

  • CAS Number: 99-14-9
  • MF: C6H8O6
  • MW: 176.124
  • Catalog: Others
  • Density: 1.6±0.1 g/cm3
  • Boiling Point: 266.4±20.0 °C at 760 mmHg
  • Melting Point: 156-161 °C(lit.)
  • Flash Point: 129.2±18.3 °C

Arteannuin L

Arteannuin L can be isolated from Artemisia annua[1]

  • CAS Number: 207446-89-7
  • MF: C15H22O3
  • MW: 250.333
  • Catalog: Others
  • Density: 1.1±0.1 g/cm3
  • Boiling Point: 420.7±38.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 178.0±19.5 °C

3,3'-Di-O-methylellagic acid 4'-glucoside

3,3'-Di-O-methylellagic acid-4'-O-β-D-glucopyranoside is a ellagic acid derivative that can be isolated from Dipentodon sinicus[1].

  • CAS Number: 51803-68-0
  • MF: C22H20O13
  • MW: 492.386
  • Catalog: Others
  • Density: 1.7±0.1 g/cm3
  • Boiling Point: 887.4±65.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 310.6±27.8 °C

Polyoxyl 40 stearate

Polyoxyl 40 stearate can be used as an excipient. Pharmaceutical excipients, or pharmaceutical auxiliaries, refer to other chemical substances used in the pharmaceutical process other than pharmaceutical ingredients. Pharmaceutical excipients generally refer to inactive ingredients in pharmaceutical preparations, which can improve the stability, solubility and processability of pharmaceutical preparations. Pharmaceutical excipients also affect the absorption, distribution, metabolism, and elimination (ADME) processes of co-administered drugs[1].

  • CAS Number: 171286-89-8
  • MF: C98H196O42
  • MW: 2046.58
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Dulcite-13C

Dulcite-13C is the 13C labeled Dulcite. Dulcite is a sugar alcohol with a slightly sweet taste which is a metabolic breakdown product of galact[1][2].

  • CAS Number: 2484171-11-9
  • MF: C513CH14O6
  • MW: 183.16
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Adenosine 5'-triphosphate(ATP)-d4 ammonium salt

Adenosine 5'-triphosphate(ATP)-d4 (ammonium salt) is the deuterium labeled Adenosine 5'-triphosphate(ATP) ammonium salt[1].

  • CAS Number: 2483831-82-7
  • MF: C10H24D4N9O13P3
  • MW: 579.33
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Dihydrorhodamine 123

Dihydrorhodamine 123 is a fluorescent probe (λex=488 nm, λem=525 nm).

  • CAS Number: 109244-58-8
  • MF: C21H18N2O3
  • MW: 346.379
  • Catalog: Dye Reagents
  • Density: 1.3±0.1 g/cm3
  • Boiling Point: 526.9±50.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 222.4±26.4 °C

Poly(ethylene glycol) tetrahydrofurfuryl ether

Poly(ethylene glycol) tetrahydrofurfuryl ether is liquid glycogen can be easily transformed into a gel system with excellent elasticity, so it can be used as a medium for dissolving water-insoluble drugs.

  • CAS Number: 31692-85-0
  • MF: (C2H4O)nC5H10O2
  • MW: 233.28
  • Catalog: Others
  • Density: 1.061g/cm3
  • Boiling Point: 256.2ºC at 760mmHg
  • Melting Point: N/A
  • Flash Point: 108.7ºC

15,16-Epoxy-12R-hydroxylabda-8(17),13(16),14-triene

15,16-Epoxy-12R-hydroxylabda-8(17),13(16),14-triene is a compound isolated from the seeds of Aframomum aulacocarpos[1].

  • CAS Number: 61597-55-5
  • MF: C20H30O2
  • MW: 302.45
  • Catalog: Others
  • Density: 1.0±0.1 g/cm3
  • Boiling Point: 328.6±9.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 152.5±18.7 °C

BDC2.5 Mimotope 1040-63

BDC2.5 Mimotope 1040-63 is a biological active peptide. (The TCR transgenic model (BDC2.5) mimitope was used in type 1 diabetes (T1D) study. T1D is an autoimmune disease in which T cells mediate damage to pancreatic islet b cells. T1D is caused by autoreactive T cell destruction of insulin-producing cells. BDC2.5 mimotope was utilized to support the study on antigen presentation of antigenic peptides to islet autoantigen-specific T cells.)

  • CAS Number: 329696-53-9
  • MF: C59H98N20O14S
  • MW: 1343.60
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Heteroclitin D

Heteroclitin D is a lignin from Kadsura medicinal plants with anti-liqid peroxidation. Heteroclitin D inhibits L-type calcium channels[1].

  • CAS Number: 140369-76-2
  • MF: C27H30O8
  • MW: 482.522
  • Catalog: Others
  • Density: 1.3±0.1 g/cm3
  • Boiling Point: 640.3±55.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 273.3±31.5 °C

Fmoc-L-Lys(Pryoc)-OH

Fmoc-L-Lys(Pryoc)-OH (N2-Fmoc-N6-[(propargyloxy)carbonyl]-L-lysine) is a click chemistry reagent containing an azide group[1].

  • CAS Number: 1584133-25-4
  • MF: C25H26N2O6
  • MW: 450.48
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

3-Mercaptopropane-1,2-diol

1-Thioglycerol is a biochemical reagent that can be used as a biological material or organic compound for life science related research.

  • CAS Number: 96-27-5
  • MF: C3H8O2S
  • MW: 108.159
  • Catalog: ATM/ATR
  • Density: 1.2±0.1 g/cm3
  • Boiling Point: 247.0±0.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 126.3±24.6 °C

Protopseudohypericin

Protopseudohypericin, a naturally occurring naphthodianthrone, is isolated from H. perforatum. Protopseudohypericin is considered to be the biosynthetic precursor of Pseudohypericin[1][2].

  • CAS Number: 54328-09-5
  • MF: C30H18O9
  • MW: 522.458
  • Catalog: Others
  • Density: 1.8±0.1 g/cm3
  • Boiling Point: 1019.3±65.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 584.0±30.8 °C

Tetrabenazine D6

Tetrabenazine D6 is the deuterium labeled Tetrabenazine, which is a VMAT-inhibitor used for treatment of hyperkinetic movement disorder.

  • CAS Number: 1392826-25-3
  • MF: C19H21D6NO3
  • MW: 323.46000
  • Catalog: Monoamine Transporter
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

1-Methyl(3,3,5,5-2H4)piperazine

N-Methylpiperazine-d4 is the deuterium labeled N-Methylpiperazine[1].

  • CAS Number: 343864-02-8
  • MF: C5H8D4N2
  • MW: 104.187
  • Catalog: Others
  • Density: 0.9±0.1 g/cm3
  • Boiling Point: 138.0±8.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 42.2±0.0 °C

BODIPY FL Verapamil hydrochloride

BODIPY FL Verapamil hydrochloride is a fluorescent dye, it can be used as a molecular probe to label tissues and cells. BODIPY FL Verapamil hydrochloride is a substrate for both ABCB1 and ABCC1[1][2].

  • CAS Number: 216571-88-9
  • MF: C41H56BClF2N4O5
  • MW: 769.17
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A