Chemsrc provides Others's classification. They are divided into Androgen Receptor, Aromatase, Estrogen Receptor/ERR, Progesterone Receptor, Thyroid Hormone Receptor, Others according to their Biological activity.


Anti-infection >
Arenavirus Bacterial CMV Enterovirus Filovirus Fungal HBV HCV HIV HSV Influenza Virus Parasite Reverse Transcriptase RSV SARS-CoV
Antibody-drug Conjugate >
ADC Cytotoxin ADC Linker Drug-Linker Conjugates for ADC PROTAC-linker Conjugate for PAC
Apoptosis >
Apoptosis Bcl-2 Family c-Myc Caspase DAPK Ferroptosis IAP MDM-2/p53 PKD RIP kinase Survivin Thymidylate Synthase TNF Receptor
Autophagy >
Autophagy LRRK2 ULK Mitophagy
Cell Cycle/DNA Damage >
Antifolate APC ATM/ATR Aurora Kinase Casein Kinase CDK Checkpoint Kinase (Chk) CRISPR/Cas9 Deubiquitinase DNA Alkylator/Crosslinker DNA-PK DNA/RNA Synthesis Eukaryotic Initiation Factor (eIF) G-quadruplex Haspin Kinase HDAC HSP IRE1 Kinesin LIM Kinase (LIMK) Microtubule/Tubulin Mps1 Nucleoside Antimetabolite/Analog p97 PAK PARP PERK Polo-like Kinase (PLK) PPAR RAD51 ROCK Sirtuin SRPK Telomerase TOPK Topoisomerase Wee1
Cytoskeleton >
Arp2/3 Complex Dynamin Gap Junction Protein Integrin Kinesin Microtubule/Tubulin Mps1 Myosin PAK
Epigenetics >
AMPK Aurora Kinase DNA Methyltransferase Epigenetic Reader Domain HDAC Histone Acetyltransferase Histone Demethylase Histone Methyltransferase JAK MicroRNA PARP PKC Sirtuin Protein Arginine Deiminase
GPCR/G Protein >
5-HT Receptor Adenosine Receptor Adenylate Cyclase Adiponectin Receptor Adrenergic Receptor Angiotensin Receptor Bombesin Receptor Bradykinin Receptor Cannabinoid Receptor CaSR CCR CGRP Receptor Cholecystokinin Receptor CRFR CXCR Dopamine Receptor EBI2/GPR183 Endothelin Receptor GHSR Glucagon Receptor Glucocorticoid Receptor GNRH Receptor GPCR19 GPR109A GPR119 GPR120 GPR139 GPR40 GPR55 GPR84 Guanylate Cyclase Histamine Receptor Imidazoline Receptor Leukotriene Receptor LPL Receptor mAChR MCHR1 (GPR24) Melatonin Receptor mGluR Motilin Receptor Neurokinin Receptor Neuropeptide Y Receptor Neurotensin Receptor Opioid Receptor Orexin Receptor (OX Receptor) Oxytocin Receptor P2Y Receptor Prostaglandin Receptor Protease-Activated Receptor (PAR) Ras RGS Protein Sigma Receptor Somatostatin Receptor TSH Receptor Urotensin Receptor Vasopressin Receptor Melanocortin Receptor
Immunology/Inflammation >
Aryl Hydrocarbon Receptor CCR Complement System COX CXCR FLAP Histamine Receptor IFNAR Interleukin Related IRAK MyD88 NO Synthase NOD-like Receptor (NLR) PD-1/PD-L1 PGE synthase Salt-inducible Kinase (SIK) SPHK STING Thrombopoietin Receptor Toll-like Receptor (TLR) Arginase
JAK/STAT Signaling >
EGFR JAK Pim STAT
MAPK/ERK Pathway >
ERK JNK KLF MAP3K MAP4K MAPKAPK2 (MK2) MEK Mixed Lineage Kinase MNK p38 MAPK Raf Ribosomal S6 Kinase (RSK)
Membrane Transporter/Ion Channel >
ATP Synthase BCRP Calcium Channel CFTR Chloride Channel CRAC Channel CRM1 EAAT2 GABA Receptor GlyT HCN Channel iGluR Monoamine Transporter Monocarboxylate Transporter Na+/Ca2+ Exchanger Na+/HCO3- Cotransporter Na+/K+ ATPase nAChR NKCC P-glycoprotein P2X Receptor Potassium Channel Proton Pump SGLT Sodium Channel TRP Channel URAT1
Metabolic Enzyme/Protease >
15-PGDH 5 alpha Reductase 5-Lipoxygenase Acetyl-CoA Carboxylase Acyltransferase Adenosine Deaminase Adenosine Kinase Aldehyde Dehydrogenase (ALDH) Aldose Reductase Aminopeptidase Angiotensin-converting Enzyme (ACE) ATGL ATP Citrate Lyase Carbonic Anhydrase Carboxypeptidase Cathepsin CETP COMT Cytochrome P450 Dipeptidyl Peptidase Dopamine β-hydroxylase E1/E2/E3 Enzyme Elastase Enolase FAAH FABP Factor Xa Farnesyl Transferase Fatty Acid Synthase (FAS) FXR Glucokinase GSNOR Gutathione S-transferase HCV Protease Hexokinase HIF/HIF Prolyl-Hydroxylase HIV Integrase HIV Protease HMG-CoA Reductase (HMGCR) HSP Indoleamine 2,3-Dioxygenase (IDO) Isocitrate Dehydrogenase (IDH) Lactate Dehydrogenase LXR MAGL Mineralocorticoid Receptor Mitochondrial Metabolism MMP Nampt NEDD8-activating Enzyme Neprilysin PAI-1 PDHK PGC-1α Phosphatase Phosphodiesterase (PDE) Phospholipase Procollagen C Proteinase Proteasome Pyruvate Kinase RAR/RXR Renin ROR Ser/Thr Protease SGK Stearoyl-CoA Desaturase (SCD) Thrombin Tryptophan Hydroxylase Tyrosinase Xanthine Oxidase
Neuronal Signaling >
5-HT Receptor AChE Adenosine Kinase Amyloid-β Beta-secretase CaMK CGRP Receptor COMT Dopamine Receptor Dopamine Transporter FAAH GABA Receptor GlyT iGluR Imidazoline Receptor mAChR Melatonin Receptor Monoamine Oxidase nAChR Neurokinin Receptor Opioid Receptor Serotonin Transporter γ-secretase
NF-κB >
NF-κB IKK Keap1-Nrf2 MALT1
PI3K/Akt/mTOR >
Akt AMPK ATM/ATR DNA-PK GSK-3 MELK mTOR PDK-1 PI3K PI4K PIKfyve PTEN
PROTAC >
PROTAC E3 Ligase Ligand-Linker Conjugate Ligand for E3 Ligase PROTAC Linker PROTAC-linker Conjugate for PAC
Protein Tyrosine Kinase/RTK >
Ack1 ALK Bcr-Abl BMX Kinase Btk c-Fms c-Kit c-Met/HGFR Discoidin Domain Receptor DYRK EGFR Ephrin Receptor FAK FGFR FLT3 IGF-1R Insulin Receptor IRAK Itk PDGFR PKA Pyk2 ROS Src Syk TAM Receptor Trk Receptor VEGFR
Stem Cell/Wnt >
Casein Kinase ERK Gli GSK-3 Hedgehog Hippo (MST) JAK Notch Oct3/4 PKA Porcupine ROCK sFRP-1 Smo STAT TGF-beta/Smad Wnt YAP β-catenin γ-secretase
TGF-beta/Smad >
TGF-beta/Smad PKC ROCK TGF-β Receptor
Vitamin D Related >
VD/VDR
Others >
Androgen Receptor Aromatase Estrogen Receptor/ERR Progesterone Receptor Thyroid Hormone Receptor Others

Binetrakin

Binetrakin (Interleukin 4 (human)) is a T lymphocyte-derived pleiotrophic cytokine that affects a variety of cell types including B cells and T cells. Binetrakin induces differentiation of naive helper T cells (Th0 cells) to Th2 cells. Binetrakin can be used for the research of many biological[1][2].

  • CAS Number: 207137-56-2
  • MF:
  • MW:
  • Catalog: Inflammation/Immunology
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Soyasaponin IV

Soyasaponin IV, isolated from the aerial parts of Glycine soya, exhibits a hepatoprotective action[1].

  • CAS Number: 108906-97-4
  • MF: C41H66O13
  • MW: 766.95500
  • Catalog: Others
  • Density: N/A
  • Boiling Point: 876.8±65.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: N/A

6-benzoyl-6-deacetylmayteine

Ebenifoline E-II (Compound 2) is a sesquiterpene alkaloid derived from Euonymus laxiflorus. Ebenifoline E-II is cytotoxic[1].

  • CAS Number: 133740-16-6
  • MF: C48H51NO18
  • MW: 929.91400
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

3-Azido-L-alanine hydrochloride

3-Azido-L-alanine hydrochloride is an aliphatic functionalized amino acid with side chain lengths of up to four carbons[1].

  • CAS Number: 1620171-64-3
  • MF: C3H7ClN4O2
  • MW: 166.57
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Nilutamide

Nilutamide (Nilandron) is a non-steroidal anti-androgen drug proposed in the treatment of metastatic prostatic carcinoma[1][2].

  • CAS Number: 63612-50-0
  • MF: C12H10F3N3O4
  • MW: 317.221
  • Catalog: Cancer
  • Density: 1.5±0.1 g/cm3
  • Boiling Point: N/A
  • Melting Point: 1490C
  • Flash Point: N/A

Vitamin U

DL-methionine methylsulfonium chloride is a naturally occurring methionine derivative. DL-methionine methylsulfonium chloride protects gastric mucosal from ethanol-induced damage[1].

  • CAS Number: 3493-12-7
  • MF: C6H14ClNO2S
  • MW: 199.699
  • Catalog: Inflammation/Immunology
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: 139ºC
  • Flash Point: N/A

methyl n-methylanthranilate

Methyl N-methylanthranilate, a terpene, is a pungent compound that can be found in Citrus reticulate Blanco leaves. Methyl N-methylanthranilate has the potential for pain research[1].

  • CAS Number: 85-91-6
  • MF: C9H11NO2
  • MW: 165.189
  • Catalog: Potassium Channel
  • Density: 1.1±0.1 g/cm3
  • Boiling Point: 252.4±13.0 °C at 760 mmHg
  • Melting Point: 17-19 °C(lit.)
  • Flash Point: 106.5±19.8 °C

s-benzyl-l-cysteinol

S-Benzyl-L-cysteinol is a cysteine derivative[1].

  • CAS Number: 85803-43-6
  • MF: C10H15NOS
  • MW: 197.29700
  • Catalog: Others
  • Density: 1.155g/cm3
  • Boiling Point: 358ºC at 760 mmHg
  • Melting Point: 42-46ºC(lit.)
  • Flash Point: >230 °F

Angelol H

Angelol H is a natural tcompound isolated from Angelica pubescens MAXIM. (Umbelliferae)[1].

  • CAS Number: 83247-73-8
  • MF: C20H24O7
  • MW: 376.400
  • Catalog: Others
  • Density: 1.3±0.1 g/cm3
  • Boiling Point: 579.1±50.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 203.1±23.6 °C

16-Methoxystrychnine

16-Methoxystrychnine is a alkaloid[1].

  • CAS Number: 5096-72-0
  • MF: C22H24N2O3
  • MW: 364.43800
  • Catalog: Others
  • Density: 1.41g/cm3
  • Boiling Point: 567.1ºC at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 296.8ºC

3,4,6-Tri-O-acetyl-D-glucal-13C

3,4,6-Tri-O-acetyl-D-glucal-13C is the 13C labeled 3,4,6-Tri-O-acetyl-D-glucal[1].

  • CAS Number: 478529-35-0
  • MF: C12H16O7
  • MW: 273.24400
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

2-Methylpiperazine-d10

2-Methylpiperazine-d10 is the deuterium labeled 2-Methylpiperazine[1].

  • CAS Number: 2363789-19-7
  • MF: C5H2D10N2
  • MW: 110.22
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

AZ 1729

AZ1729 is a novel direct, positive allosteric modulator of fatty acid receptor FFA2 (pEC50=6.9), selectively activates Gi signaling but lacks the capacity to activate FFA2 Gq/G11-mediated signaling pathways; produces stimulation of [35S]GTPγS binding with pEC50 7.23, inhibits β-adrenoreceptor agonist-promoted lipolysis in primary mouse adipocytes and promotes chemotaxis of isolated human neutrophils.

  • CAS Number: 2016864-46-1
  • MF: C18H16FN5OS
  • MW: 369.418
  • Catalog: Metabolic Disease
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Mefox

Mefox is a degradation product of folic acid (HY-16637)[1].

  • CAS Number: 79573-48-1
  • MF: C20H23N7O7
  • MW: 473.44
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Ro 5-3335

Ro5-3335, a benzodiazepine, acts as an inhibitor of core binding factor (CBF) leukemia. Ro5-3335 is a RUNX1-CBFβ interaction inhibitor that represses RUNX1/CBFB-dependent transactivation[1].

  • CAS Number: 30195-30-3
  • MF: C13H10ClN3O
  • MW: 259.69100
  • Catalog: Others
  • Density: 1.46g/cm3
  • Boiling Point: 501.6ºC at 760mmHg
  • Melting Point: 256 °C (分解)
  • Flash Point: 257.1ºC

Rocagloic acid

Rocagloic acid is a racaglamide derivative isolated from the fruits of Amoora cucullata with potent cytotoxicity[1].

  • CAS Number: 190385-15-0
  • MF: C27H26O8
  • MW: 478.49
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Cyclo(D-Ala-L-Pro)

Cyclo(D-Ala-L-Pro) is a cyclodipeptide[1].

  • CAS Number: 36238-64-9
  • MF: C8H12N2O2
  • MW: 168.19300
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

LGD-3303

LGD-3303 is a selective androgen receptor modulator (SARM).

  • CAS Number: 917891-35-1
  • MF: C16H14ClF3N2O
  • MW: 342.74300
  • Catalog: Endocrinology
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Cnidioside B

Cnidioside B is a glycoside compound, which can be isolated from Leptothyrsa sprucei, C. monnieri and the ripe fruit of Cnidium monieri[1][2][3].

  • CAS Number: 141896-54-0
  • MF: C18H22O10
  • MW: 398.36
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

8-Azanebularine

8-Azanebularine, a compound with hydrogen in place of the C6 amino group, inhibits the ADAR2 reaction at high concentrations (IC50=15 mM). 8-Azanebularine is incorporated into an RNA structure recognized by human ADAR2 results in high-affinity binding (KD=2 nM). 8-Azanebularine can be used for the research of ADAR-catalyzed RNA-editing reaction[1].

  • CAS Number: 38874-46-3
  • MF: C9H11N5O4
  • MW: 253.21500
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

ER degrader 5

ER degrader 5 is a potent estrogen receptor (ER) degrader. ER degrader 5 shows anti-proliferation activity. ER degrader 5 can be used for the research of breast cancer[1].

  • CAS Number: 2913192-47-7
  • MF: C26H18F2O4S
  • MW: 464.48
  • Catalog: Cancer
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Trinexapac-ethyl

Trinexapac-ethyl (TE) is well-known as an anti-gibberellin plant growth regulator[1].

  • CAS Number: 95266-40-3
  • MF: C13H16O5
  • MW: 252.263
  • Catalog: Endocrinology
  • Density: 1.4±0.1 g/cm3
  • Boiling Point: 399.4±42.0 °C at 760 mmHg
  • Melting Point: 32-36ºC
  • Flash Point: 150.8±21.4 °C

N-Hydroxypipecolic acid potassium

N-Hydroxypipecolic acid potassium (1-Hydroxy-2-piperidinecarboxylic acid potassium), a plant metabolite and a systemic acquired resistance (SAR) regulator, orchestrates SAR establishment in concert with the immune signal salicylic acid. N-Hydroxypipecolic acid potassium accumulates systemically in the plant foliage in response to pathogen attack. N-Hydroxypipecolic acid potassium induces SAR to bacterial and oomycete infection[1][2][3].

  • CAS Number: 2253632-01-6
  • MF: C6H10KNO3
  • MW: 183.25
  • Catalog: Inflammation/Immunology
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

2,3,5,6-Tetramethoxyaporphine

2,3,5,6-Tetramethoxyaporphine is an antitussive agent, a medicinally valuable benzyl isoquinoline alkaloid. 2,3,5,6-Tetramethoxyaporphine can be isolated from the yellow hornpoppy, Glaucium flavum Cr. (Fam. Papaveraceae)[1][2].

  • CAS Number: 5630-11-5
  • MF: C21H25NO4
  • MW: 355.42800
  • Catalog: Others
  • Density: 1.166g/cm3
  • Boiling Point: 487ºC at 760 mmHg
  • Melting Point: 119ºC
  • Flash Point: 140.2ºC

TA-7552

TA-7552 is a potent cholesterol-lowering agent.

  • CAS Number: 104756-72-1
  • MF: C25H26O10
  • MW: 486.46800
  • Catalog: Cardiovascular Disease
  • Density: 1.269g/cm3
  • Boiling Point: 592.3ºC at 760mmHg
  • Melting Point: N/A
  • Flash Point: 195ºC

(2S)-Gemcitabine-13C,15N2 hydrochloride

(2S)-Gemcitabine-13C,15N2 (hydrochloride) is the 13C and 15N labeled (2S)-Gemcitabine hydrochloride[1].

  • CAS Number: 1262897-74-4
  • MF: C813CH12ClF2N15N2O4
  • MW: 302.639
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Leucocrystal violet

Leucocrystal violet is a triphenylmethane dye which can be used to detect antimony in environmental and biological samples using spectrophotometric techniques.

  • CAS Number: 603-48-5
  • MF: C25H31N3
  • MW: 373.534
  • Catalog: Dye Reagents
  • Density: 1.1±0.1 g/cm3
  • Boiling Point: 529.8±50.0 °C at 760 mmHg
  • Melting Point: 175-177 °C(lit.)
  • Flash Point: 281.8±20.7 °C

Sarcosine hydrochloride

2-(Methylamino)acetic acid hydrochloride is a Glycine (HY-Y0966) derivative[1].

  • CAS Number: 637-96-7
  • MF: C3H8ClNO2
  • MW: 125.554
  • Catalog: Others
  • Density: 1.48 g/cm3
  • Boiling Point: 195.1ºC at 760 mmHg
  • Melting Point: 173-175 °C(lit.)
  • Flash Point: 71.8ºC

Mitumomab

Mitumomab is an anti-idiotypic mouse IgG2b monoclonal antibody that mimics the ganglioside GD3. Mitumomab can be used for the research of small-cell lung carcinoma[1].

  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Phenazoviridin

Phenazoviridin is a free radical scavenger. Phenazoviridin shows strong inhibitory activity against lipid peroxidation in rat brain homogenate and exhibits antihypoxic activity in mice[1].

  • CAS Number: 155233-15-1
  • MF: C24H26N2O6
  • MW: 438.47300
  • Catalog: Cancer
  • Density: 1.38g/cm3
  • Boiling Point: 661.1ºC at 760mmHg
  • Melting Point: N/A
  • Flash Point: 353.6ºC