Chemsrc provides Others's classification, including all related biologically active compounds cover the research fields of cancer, neuroscience, immunology and other popular diseases, etc.


Anti-infection >
Arenavirus Bacterial CMV Enterovirus Filovirus Fungal HBV HCV HIV HSV Influenza Virus Parasite Reverse Transcriptase RSV SARS-CoV
Antibody-drug Conjugate >
ADC Cytotoxin ADC Linker Drug-Linker Conjugates for ADC PROTAC-linker Conjugate for PAC
Apoptosis >
Apoptosis Bcl-2 Family c-Myc Caspase DAPK Ferroptosis IAP MDM-2/p53 PKD RIP kinase Survivin Thymidylate Synthase TNF Receptor
Autophagy >
Autophagy LRRK2 ULK Mitophagy
Cell Cycle/DNA Damage >
Antifolate APC ATM/ATR Aurora Kinase Casein Kinase CDK Checkpoint Kinase (Chk) CRISPR/Cas9 Deubiquitinase DNA Alkylator/Crosslinker DNA-PK DNA/RNA Synthesis Eukaryotic Initiation Factor (eIF) G-quadruplex Haspin Kinase HDAC HSP IRE1 Kinesin LIM Kinase (LIMK) Microtubule/Tubulin Mps1 Nucleoside Antimetabolite/Analog p97 PAK PARP PERK Polo-like Kinase (PLK) PPAR RAD51 ROCK Sirtuin SRPK Telomerase TOPK Topoisomerase Wee1
Cytoskeleton >
Arp2/3 Complex Dynamin Gap Junction Protein Integrin Kinesin Microtubule/Tubulin Mps1 Myosin PAK
Epigenetics >
AMPK Aurora Kinase DNA Methyltransferase Epigenetic Reader Domain HDAC Histone Acetyltransferase Histone Demethylase Histone Methyltransferase JAK MicroRNA PARP PKC Sirtuin Protein Arginine Deiminase
GPCR/G Protein >
5-HT Receptor Adenosine Receptor Adenylate Cyclase Adiponectin Receptor Adrenergic Receptor Angiotensin Receptor Bombesin Receptor Bradykinin Receptor Cannabinoid Receptor CaSR CCR CGRP Receptor Cholecystokinin Receptor CRFR CXCR Dopamine Receptor EBI2/GPR183 Endothelin Receptor GHSR Glucagon Receptor Glucocorticoid Receptor GNRH Receptor GPCR19 GPR109A GPR119 GPR120 GPR139 GPR40 GPR55 GPR84 Guanylate Cyclase Histamine Receptor Imidazoline Receptor Leukotriene Receptor LPL Receptor mAChR MCHR1 (GPR24) Melatonin Receptor mGluR Motilin Receptor Neurokinin Receptor Neuropeptide Y Receptor Neurotensin Receptor Opioid Receptor Orexin Receptor (OX Receptor) Oxytocin Receptor P2Y Receptor Prostaglandin Receptor Protease-Activated Receptor (PAR) Ras RGS Protein Sigma Receptor Somatostatin Receptor TSH Receptor Urotensin Receptor Vasopressin Receptor Melanocortin Receptor
Immunology/Inflammation >
Aryl Hydrocarbon Receptor CCR Complement System COX CXCR FLAP Histamine Receptor IFNAR Interleukin Related IRAK MyD88 NO Synthase NOD-like Receptor (NLR) PD-1/PD-L1 PGE synthase Salt-inducible Kinase (SIK) SPHK STING Thrombopoietin Receptor Toll-like Receptor (TLR) Arginase
JAK/STAT Signaling >
EGFR JAK Pim STAT
MAPK/ERK Pathway >
ERK JNK KLF MAP3K MAP4K MAPKAPK2 (MK2) MEK Mixed Lineage Kinase MNK p38 MAPK Raf Ribosomal S6 Kinase (RSK)
Membrane Transporter/Ion Channel >
ATP Synthase BCRP Calcium Channel CFTR Chloride Channel CRAC Channel CRM1 EAAT2 GABA Receptor GlyT HCN Channel iGluR Monoamine Transporter Monocarboxylate Transporter Na+/Ca2+ Exchanger Na+/HCO3- Cotransporter Na+/K+ ATPase nAChR NKCC P-glycoprotein P2X Receptor Potassium Channel Proton Pump SGLT Sodium Channel TRP Channel URAT1
Metabolic Enzyme/Protease >
15-PGDH 5 alpha Reductase 5-Lipoxygenase Acetyl-CoA Carboxylase Acyltransferase Adenosine Deaminase Adenosine Kinase Aldehyde Dehydrogenase (ALDH) Aldose Reductase Aminopeptidase Angiotensin-converting Enzyme (ACE) ATGL ATP Citrate Lyase Carbonic Anhydrase Carboxypeptidase Cathepsin CETP COMT Cytochrome P450 Dipeptidyl Peptidase Dopamine β-hydroxylase E1/E2/E3 Enzyme Elastase Enolase FAAH FABP Factor Xa Farnesyl Transferase Fatty Acid Synthase (FAS) FXR Glucokinase GSNOR Gutathione S-transferase HCV Protease Hexokinase HIF/HIF Prolyl-Hydroxylase HIV Integrase HIV Protease HMG-CoA Reductase (HMGCR) HSP Indoleamine 2,3-Dioxygenase (IDO) Isocitrate Dehydrogenase (IDH) Lactate Dehydrogenase LXR MAGL Mineralocorticoid Receptor Mitochondrial Metabolism MMP Nampt NEDD8-activating Enzyme Neprilysin PAI-1 PDHK PGC-1α Phosphatase Phosphodiesterase (PDE) Phospholipase Procollagen C Proteinase Proteasome Pyruvate Kinase RAR/RXR Renin ROR Ser/Thr Protease SGK Stearoyl-CoA Desaturase (SCD) Thrombin Tryptophan Hydroxylase Tyrosinase Xanthine Oxidase
Neuronal Signaling >
5-HT Receptor AChE Adenosine Kinase Amyloid-β Beta-secretase CaMK CGRP Receptor COMT Dopamine Receptor Dopamine Transporter FAAH GABA Receptor GlyT iGluR Imidazoline Receptor mAChR Melatonin Receptor Monoamine Oxidase nAChR Neurokinin Receptor Opioid Receptor Serotonin Transporter γ-secretase
NF-κB >
NF-κB IKK Keap1-Nrf2 MALT1
PI3K/Akt/mTOR >
Akt AMPK ATM/ATR DNA-PK GSK-3 MELK mTOR PDK-1 PI3K PI4K PIKfyve PTEN
PROTAC >
PROTAC E3 Ligase Ligand-Linker Conjugate Ligand for E3 Ligase PROTAC Linker PROTAC-linker Conjugate for PAC
Protein Tyrosine Kinase/RTK >
Ack1 ALK Bcr-Abl BMX Kinase Btk c-Fms c-Kit c-Met/HGFR Discoidin Domain Receptor DYRK EGFR Ephrin Receptor FAK FGFR FLT3 IGF-1R Insulin Receptor IRAK Itk PDGFR PKA Pyk2 ROS Src Syk TAM Receptor Trk Receptor VEGFR
Stem Cell/Wnt >
Casein Kinase ERK Gli GSK-3 Hedgehog Hippo (MST) JAK Notch Oct3/4 PKA Porcupine ROCK sFRP-1 Smo STAT TGF-beta/Smad Wnt YAP β-catenin γ-secretase
TGF-beta/Smad >
TGF-beta/Smad PKC ROCK TGF-β Receptor
Vitamin D Related >
VD/VDR
Others >
Androgen Receptor Aromatase Estrogen Receptor/ERR Progesterone Receptor Thyroid Hormone Receptor Others

2-Pyridinecarbohydrazide

2-Pyridinecarbohydrazide is a building block extensively used in various fields of synthesis[1].

  • CAS Number: 1452-63-7
  • MF: C6H7N3O
  • MW: 137.139
  • Catalog: Others
  • Density: 1.2±0.1 g/cm3
  • Boiling Point: N/A
  • Melting Point: 100°C
  • Flash Point: N/A

3-(Methyl-nitrosoamino)propionitrile-d3

3-(Methyl-nitrosoamino)propionitrile-d3 is the deuterium labeled 3-(Methyl-nitrosoamino)propionitrile[1].

  • CAS Number: 1329834-39-0
  • MF: C4H4D3N3O
  • MW: 116.14
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Astressin TFA

Astressin is a potent corticotropin releasing factor (CRF) antagonist.

  • CAS Number: 170809-51-5
  • MF: C161H269N49O42
  • MW: 3563.16000
  • Catalog: Peptides
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Biotin-16-dUTP

Biotin-16-dUTP is a fluorescent substitute of dTTP.

  • CAS Number: 86303-26-6
  • MF: C32H52N7O18P3S
  • MW: 947.78
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

3FAx-Neu5Ac

3FAx-Neu5Ac (compound 8), a Sialic acid peracetylated analog, is a sialyltransferase inhibitor. 3FAx-Neu5Ac substantially reduces expression of the sialylated ligand sialyl Lewis X on myeloid cells[1].

  • CAS Number: 117405-58-0
  • MF: C22H30FNO14
  • MW: 551.47
  • Catalog: Metabolic Disease
  • Density: 1.4±0.1 g/cm3
  • Boiling Point: 606.3±55.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 320.5±31.5 °C

Telimomab aritox

Telimomab aritox (T101-ricin A chain immunotoxin) is a mouse monoclonal antibody that linked to the A chain of the ricin protein. Telimomab aritox can be used as an immunosuppressive agent[1].

  • CAS Number: 117305-33-6
  • MF:
  • MW:
  • Catalog: Inflammation/Immunology
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

A 971432

A-971432 is a potent, selective and orally active sphingosine-1-phosphate (S1P) receptor 5 agonist with IC50s of .362, >10, 0.006 µM for S1P1, S1P3, S1P5 respectively. A-971432 protects blood–brain barrier (BBB) homeostasis. A-971432 reverses age-related cognitive decline. A-971432 has the potential for the research of alzheimer’s disease or multiple sclerosis [1][2].

  • CAS Number: 1240308-45-5
  • MF: C18H17Cl2NO3
  • MW: 366.24
  • Catalog: Neurological Disease
  • Density: 1.4±0.1 g/cm3
  • Boiling Point: 520.0±50.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 268.3±30.1 °C

Lactoferrin (322-329) (human) trifluoroacetate salt

Lactoferrin (322-329) (human) is a polypeptide that can be found by peptide screening. Peptide screening is a research tool that pools active peptides primarily by immunoassay. Peptide screening can be used for protein interaction, functional analysis, epitope screening, especially in the field of agent research and development[1].

  • CAS Number: 496808-32-3
  • MF: C35H53N9O12
  • MW: 791.85
  • Catalog: Others
  • Density: 1.3±0.1 g/cm3
  • Boiling Point: 1318.8±65.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 751.4±34.3 °C

Luciferase, firefly

Luciferase, firefly is the light-emitting enzyme responsible for the bioluminescence of fireflies and click beetles.

  • CAS Number: 61970-00-1
  • MF: C19H20N2O4
  • MW:
  • Catalog: Peptides
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

1-palmitoyl-d31-2-oleoyl-sn-glycero-3-phosphoinositol (ammonium salt)

1-Palmitoyl-2-oleoyl-sn-glycero-3-phosphoinositol-d31 (ammonium) is deuterium labeled 1-Palmitoyl-2-oleoyl-sn-glycero-3-phosphoinositol (ammonium).

  • CAS Number: 799812-61-6
  • MF: C43H53D31NO13P
  • MW: 885.291
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Boc-N-Me-Ser-OH

Boc-N-Me-Ser-OH is a serine derivative[1].

  • CAS Number: 101772-29-6
  • MF: C9H17NO5
  • MW: 219.235
  • Catalog: Others
  • Density: 1.2±0.1 g/cm3
  • Boiling Point: 353.2±42.0 °C at 760 mmHg
  • Melting Point: 83-87ºC
  • Flash Point: 167.4±27.9 °C

(R)-2-Amino-3-(pyridin-3-yl)propanoic acid hydrochloride

H-3-D-Pal-OH.HCl is an alanine derivative[1].

  • CAS Number: 350228-35-2
  • MF: C8H11ClN2O2
  • MW: 202.63800
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Vitexdoin A

Vitexdoin A is a nitric oxide scavenging lignin. Vitexdoin A inhibits NO production with an IC50 of 0.38 μM in LPS (HY-D1056)-stimulated RAW 264.7 cells[1].

  • CAS Number: 1186021-77-1
  • MF: C19H18O6
  • MW: 342.34
  • Catalog: Inflammation/Immunology
  • Density: 1.5±0.1 g/cm3
  • Boiling Point: 612.7±55.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 224.2±25.0 °C

(R)-2-(6-((2’,6’-Dimethyl-4’-(3-(Methylsulfonyl)Propoxy)-[1,1’-Biphenyl]-3-Yl)Methoxy)-2,3-Dihydrobenzofuran-3-Yl)Acetic Acid

(R)-Fasiglifam is the inactive isomer of Fasiglifam (HY-10480), and can be used as an experimental control. Fasiglifam (TAK-875) is a potent, selective and orally bioavailable GPR40 agonist with EC50 of 72 nM.

  • CAS Number: 1234474-57-7
  • MF: C29H32O7S
  • MW: 524.63
  • Catalog: Metabolic Disease
  • Density: 1.3±0.1 g/cm3
  • Boiling Point: 739.1±60.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 400.8±32.9 °C

UDP-β-D-glucose disodium

UDP-β-D-glucose disodium is a the stereoisomer of UDP-α-D-glucose. UDP-β-D-glucose disodium is an oligosaccharide that can be used to synthesize glycoproteins and glycolipids. UDP-β-D-glucose disodium can be used as a substrate[1].

  • CAS Number: 7333-33-7
  • MF: C15H22N2Na2O17P2
  • MW: 610.27
  • Catalog: Metabolic Disease
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Methyl L-phenylalaninate hydrochloride

H-Phe-OMe.hydrochloride is a phenylalanine derivative[1].

  • CAS Number: 7524-50-7
  • MF: C10H14ClNO2
  • MW: 215.677
  • Catalog: Others
  • Density: N/A
  • Boiling Point: 264.2ºC at 760 mmHg
  • Melting Point: 156-160ºC
  • Flash Point: 126ºC

N-Formyl-Met-Ala-Ser

N-Formyl-Met-Ala-Ser is a peptide, binds to formyl peptide receptors on neutrophils.

  • CAS Number: 17351-32-5
  • MF: C12H21N3O6S
  • MW: 335.38
  • Catalog: Inflammation/Immunology
  • Density: 1.146g/cm3
  • Boiling Point: 303.7ºC at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 137.5ºC

Lutein

Lutein is a carotenoid with reported anti-inflammatory properties. A large body of evidence shows that lutein has several beneficial effects, especially on eye health[1].

  • CAS Number: 127-40-2
  • MF: C40H56O2
  • MW: 568.871
  • Catalog: Apoptosis
  • Density: 1.0±0.1 g/cm3
  • Boiling Point: 702.3±60.0 °C at 760 mmHg
  • Melting Point: 183℃
  • Flash Point: 269.1±27.5 °C

C15 Ceramide-1-phosphate-d7

C15 Ceramide-1-phosphate-d7 is deuterium labeled C15 Ceramide-1-phosphate.

  • CAS Number: 2315262-27-0
  • MF: C33H62D7N2O6P
  • MW: 627.93
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

(+)-D-3-Carene

(+)-3-Carene, a bicyclic monoterpene, is one of the major components of the pine tree essential oils. (+)-3-Carene is a (+)-enantiomer of 3-Carene[1].

  • CAS Number: 498-15-7
  • MF: C10H16
  • MW: 136.23
  • Catalog: Inflammation/Immunology
  • Density: 0.865
  • Boiling Point: 170-172ºC
  • Melting Point: N/A
  • Flash Point: 55ºC

Tributyl citrate

Tributyl citrate is a citric acid ester. Tributyl citrate can be used as an excipient, such as plasticizer. Pharmaceutical excipients, or pharmaceutical auxiliaries, refer to other chemical substances used in the pharmaceutical process other than pharmaceutical ingredients. Pharmaceutical excipients generally refer to inactive ingredients in pharmaceutical preparations, which can improve the stability, solubility and processability of pharmaceutical preparations. Pharmaceutical excipients also affect the absorption, distribution, metabolism, and elimination (ADME) processes of co-administered drugs[1][2].

  • CAS Number: 77-94-1
  • MF: C18H32O7
  • MW: 360.45
  • Catalog: Others
  • Density: 1.1±0.1 g/cm3
  • Boiling Point: 389.8±9.0 °C at 760 mmHg
  • Melting Point: ≥300 °C(lit.)
  • Flash Point: 120.7±12.2 °C

D-threo-PPMP

D-threo-PPMP is a potent inhibitor of glucosylceramide (GlcCer) synthase. D-threo-PPMP can block karyokinesis and reduce cyst production[1][2].

  • CAS Number: 139889-53-5
  • MF: C29H50N2O3
  • MW: 474.72
  • Catalog: Neurological Disease
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Rabacfosadine succinate

Rabacfosadine (GS-9219) succinate, a novel proagent of the nucleotide analogue PMEG, is designed as a cytotoxic agent that preferentially targets lymphoid cells[1].

  • CAS Number: 1431856-99-3
  • MF: C25H41N8O10P
  • MW: 644.61400
  • Catalog: Cancer
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

8-Hydroxyquinoline

8-Hydroxyquinoline is a monoprotic bidentate chelating agent, exhibits antiseptic, disinfectant, and pesticide properties, functioning as a transcription inhibitor.

  • CAS Number: 148-24-3
  • MF: C9H7NO
  • MW: 145.158
  • Catalog: Others
  • Density: 1.3±0.1 g/cm3
  • Boiling Point: 267.0±0.0 °C at 760 mmHg
  • Melting Point: 70-73 °C(lit.)
  • Flash Point: 143.1±20.4 °C

Repaglinide D5

Repaglinide D5 (AG-EE 623ZW D5) is deuterium labeled Repaglinide. Repaglinide is an insulin secretagogue for the treatment of type-2 diabetes mellitus[1].

  • CAS Number: 1217709-85-7
  • MF: C27H31D5N2O4
  • MW: 457.61700
  • Catalog: Metabolic Disease
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Ilexoside D

Ilexoside D is isolated from the roots of Ilex pubescens Hook. et Arn. Ilexoside D has the anti-tissue factor activity as well as the antithrombotic activity[1].

  • CAS Number: 109008-27-7
  • MF: C41H66O13
  • MW: 766.95500
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Influenza NP (311-325)

Influenza NP (311-325) is a biological active peptide. (This peptide is amino acids 311 to 325 fragment of the influenza virus nucleoprotein (NP). This bona fide MHC class II restricted epitope from influenza virus was used to study the host immunoresponse during the infection. This peptide elicits the strongest gamma interferon (IFN-gamma) production in the intracellular cytokine assays. It does not stimulate CD8 T-cells in mice.Pyroglutamyl (pGlu) peptides may spontaneously form when either Glutamine (Q) or Glutamic acid (E) is located at the sequence N-terminus. The conversion of Q or E to pGlu is a natural occurrence and in general it is believed that the hydrophobic γ-lactam ring of pGlu may play a role in peptide stability against gastrointestinal proteases. Pyroglutamyl peptides are therefore considered a normal subset of such peptides and are included as part of the peptide purity during HPLC analysis.)

  • CAS Number: 1225029-27-5
  • MF: C78H124N24O23
  • MW: 1765.97
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Fmoc-DAP-N3

Fmoc-DAP-N3 is a click chemistry reagent containing an azide group. Fmoc-DAP-N3 is a short, linear spacer molecule with Fmoc protected amino function. Fmoc-DAP-N3 can be used in click conjugation and amid bond formation either with small molecules or for bioconjugation with proteins and antibodies[1].

  • CAS Number: 1021422-85-4
  • MF: C18H18N4O2
  • MW: 322.36
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Histone H2b(29-35)

Histone H2b(29-35) is a synthetic heptapeptide that used as a substrate for cGMP-dependant kinase[1].

  • CAS Number: 71937-87-6
  • MF: C38H74N18O11
  • MW: 959.11
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Mearnsitrin

Mearnsitrin (compound 8) is a flavonol that can be isolated from methanolic extract Myrcia multiflora DC[1].

  • CAS Number: 30484-88-9
  • MF: C22H22O12
  • MW: 478.40300
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A