Chemsrc provides Others's classification, including all related biologically active compounds cover the research fields of cancer, neuroscience, immunology and other popular diseases, etc.


Anti-infection >
Arenavirus Bacterial CMV Enterovirus Filovirus Fungal HBV HCV HIV HSV Influenza Virus Parasite Reverse Transcriptase RSV SARS-CoV
Antibody-drug Conjugate >
ADC Cytotoxin ADC Linker Drug-Linker Conjugates for ADC PROTAC-linker Conjugate for PAC
Apoptosis >
Apoptosis Bcl-2 Family c-Myc Caspase DAPK Ferroptosis IAP MDM-2/p53 PKD RIP kinase Survivin Thymidylate Synthase TNF Receptor
Autophagy >
Autophagy LRRK2 ULK Mitophagy
Cell Cycle/DNA Damage >
Antifolate APC ATM/ATR Aurora Kinase Casein Kinase CDK Checkpoint Kinase (Chk) CRISPR/Cas9 Deubiquitinase DNA Alkylator/Crosslinker DNA-PK DNA/RNA Synthesis Eukaryotic Initiation Factor (eIF) G-quadruplex Haspin Kinase HDAC HSP IRE1 Kinesin LIM Kinase (LIMK) Microtubule/Tubulin Mps1 Nucleoside Antimetabolite/Analog p97 PAK PARP PERK Polo-like Kinase (PLK) PPAR RAD51 ROCK Sirtuin SRPK Telomerase TOPK Topoisomerase Wee1
Cytoskeleton >
Arp2/3 Complex Dynamin Gap Junction Protein Integrin Kinesin Microtubule/Tubulin Mps1 Myosin PAK
Epigenetics >
AMPK Aurora Kinase DNA Methyltransferase Epigenetic Reader Domain HDAC Histone Acetyltransferase Histone Demethylase Histone Methyltransferase JAK MicroRNA PARP PKC Sirtuin Protein Arginine Deiminase
GPCR/G Protein >
5-HT Receptor Adenosine Receptor Adenylate Cyclase Adiponectin Receptor Adrenergic Receptor Angiotensin Receptor Bombesin Receptor Bradykinin Receptor Cannabinoid Receptor CaSR CCR CGRP Receptor Cholecystokinin Receptor CRFR CXCR Dopamine Receptor EBI2/GPR183 Endothelin Receptor GHSR Glucagon Receptor Glucocorticoid Receptor GNRH Receptor GPCR19 GPR109A GPR119 GPR120 GPR139 GPR40 GPR55 GPR84 Guanylate Cyclase Histamine Receptor Imidazoline Receptor Leukotriene Receptor LPL Receptor mAChR MCHR1 (GPR24) Melatonin Receptor mGluR Motilin Receptor Neurokinin Receptor Neuropeptide Y Receptor Neurotensin Receptor Opioid Receptor Orexin Receptor (OX Receptor) Oxytocin Receptor P2Y Receptor Prostaglandin Receptor Protease-Activated Receptor (PAR) Ras RGS Protein Sigma Receptor Somatostatin Receptor TSH Receptor Urotensin Receptor Vasopressin Receptor Melanocortin Receptor
Immunology/Inflammation >
Aryl Hydrocarbon Receptor CCR Complement System COX CXCR FLAP Histamine Receptor IFNAR Interleukin Related IRAK MyD88 NO Synthase NOD-like Receptor (NLR) PD-1/PD-L1 PGE synthase Salt-inducible Kinase (SIK) SPHK STING Thrombopoietin Receptor Toll-like Receptor (TLR) Arginase
JAK/STAT Signaling >
EGFR JAK Pim STAT
MAPK/ERK Pathway >
ERK JNK KLF MAP3K MAP4K MAPKAPK2 (MK2) MEK Mixed Lineage Kinase MNK p38 MAPK Raf Ribosomal S6 Kinase (RSK)
Membrane Transporter/Ion Channel >
ATP Synthase BCRP Calcium Channel CFTR Chloride Channel CRAC Channel CRM1 EAAT2 GABA Receptor GlyT HCN Channel iGluR Monoamine Transporter Monocarboxylate Transporter Na+/Ca2+ Exchanger Na+/HCO3- Cotransporter Na+/K+ ATPase nAChR NKCC P-glycoprotein P2X Receptor Potassium Channel Proton Pump SGLT Sodium Channel TRP Channel URAT1
Metabolic Enzyme/Protease >
15-PGDH 5 alpha Reductase 5-Lipoxygenase Acetyl-CoA Carboxylase Acyltransferase Adenosine Deaminase Adenosine Kinase Aldehyde Dehydrogenase (ALDH) Aldose Reductase Aminopeptidase Angiotensin-converting Enzyme (ACE) ATGL ATP Citrate Lyase Carbonic Anhydrase Carboxypeptidase Cathepsin CETP COMT Cytochrome P450 Dipeptidyl Peptidase Dopamine β-hydroxylase E1/E2/E3 Enzyme Elastase Enolase FAAH FABP Factor Xa Farnesyl Transferase Fatty Acid Synthase (FAS) FXR Glucokinase GSNOR Gutathione S-transferase HCV Protease Hexokinase HIF/HIF Prolyl-Hydroxylase HIV Integrase HIV Protease HMG-CoA Reductase (HMGCR) HSP Indoleamine 2,3-Dioxygenase (IDO) Isocitrate Dehydrogenase (IDH) Lactate Dehydrogenase LXR MAGL Mineralocorticoid Receptor Mitochondrial Metabolism MMP Nampt NEDD8-activating Enzyme Neprilysin PAI-1 PDHK PGC-1α Phosphatase Phosphodiesterase (PDE) Phospholipase Procollagen C Proteinase Proteasome Pyruvate Kinase RAR/RXR Renin ROR Ser/Thr Protease SGK Stearoyl-CoA Desaturase (SCD) Thrombin Tryptophan Hydroxylase Tyrosinase Xanthine Oxidase
Neuronal Signaling >
5-HT Receptor AChE Adenosine Kinase Amyloid-β Beta-secretase CaMK CGRP Receptor COMT Dopamine Receptor Dopamine Transporter FAAH GABA Receptor GlyT iGluR Imidazoline Receptor mAChR Melatonin Receptor Monoamine Oxidase nAChR Neurokinin Receptor Opioid Receptor Serotonin Transporter γ-secretase
NF-κB >
NF-κB IKK Keap1-Nrf2 MALT1
PI3K/Akt/mTOR >
Akt AMPK ATM/ATR DNA-PK GSK-3 MELK mTOR PDK-1 PI3K PI4K PIKfyve PTEN
PROTAC >
PROTAC E3 Ligase Ligand-Linker Conjugate Ligand for E3 Ligase PROTAC Linker PROTAC-linker Conjugate for PAC
Protein Tyrosine Kinase/RTK >
Ack1 ALK Bcr-Abl BMX Kinase Btk c-Fms c-Kit c-Met/HGFR Discoidin Domain Receptor DYRK EGFR Ephrin Receptor FAK FGFR FLT3 IGF-1R Insulin Receptor IRAK Itk PDGFR PKA Pyk2 ROS Src Syk TAM Receptor Trk Receptor VEGFR
Stem Cell/Wnt >
Casein Kinase ERK Gli GSK-3 Hedgehog Hippo (MST) JAK Notch Oct3/4 PKA Porcupine ROCK sFRP-1 Smo STAT TGF-beta/Smad Wnt YAP β-catenin γ-secretase
TGF-beta/Smad >
TGF-beta/Smad PKC ROCK TGF-β Receptor
Vitamin D Related >
VD/VDR
Others >
Androgen Receptor Aromatase Estrogen Receptor/ERR Progesterone Receptor Thyroid Hormone Receptor Others

Imazamox

Imazamox is an imidazolinone (IMI) herbicides, inhibition of the biosynthesis of acetohydroxyacid synthase, which would then inhibit plant growth and ultimately lead to plant death.increase the GST (The glutathione-S-transferase) activity.in vivo: Half-life of imazamox in the soil ranges from 1 to 3 months exhibit low mammalian toxicity. [1] plants are treated with imazamox (250 μM) in the nutrient solution and harvested 7 days after. Imazamox is mainly accumulated inV. sativa, six fold higher than those detected in P.vulgaris. [2]

  • CAS Number: 114311-32-9
  • MF: C15H19N3O4
  • MW: 305.329
  • Catalog: Others
  • Density: 1.3±0.1 g/cm3
  • Boiling Point: N/A
  • Melting Point: 166-167°C
  • Flash Point: N/A

Compound 919278

LTβR-IN-1 is a potent, selective lymphotoxin β receptor (LTβR) inhibitor with an IC50 of 10 μM. LTβR-IN-1 is potent in TWEAK-stimulated p52 translocation assays with an IC50 of 10 μM and did not alter TNF-α–induced p65 nuclear translocation[1].

  • CAS Number: 2189366-77-4
  • MF: C18H16N4O2
  • MW: 320.35
  • Catalog: Metabolic Disease
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Indigo carmine

Indigo carmine is an efficient reagent for the determination of ozone by chemlluminescence (CL)[1].

  • CAS Number: 860-22-0
  • MF: C16H8N2Na2O8S2
  • MW: 466.353
  • Catalog: Others
  • Density: 1.01 g/mL at 20 °C
  • Boiling Point: N/A
  • Melting Point: >300°C
  • Flash Point: N/A

Ac-Phe-Phe-OH

Ac-Phe-Phe-OH is a negatively charged analogue of the diphenylalanine peptide that forms large aggregates when combined with the NH2-Phe-Phe-OH peptide[1].

  • CAS Number: 10030-31-6
  • MF: C20H22N2O4
  • MW: 354.40
  • Catalog: Others
  • Density: 1.225g/cm3
  • Boiling Point: 692.3ºC at 760mmHg
  • Melting Point: N/A
  • Flash Point: 372.5ºC

Fmoc-D-Ala-OH

Fmoc-D-Ala-OH is an alanine derivative[1].

  • CAS Number: 79990-15-1
  • MF: C18H17NO4
  • MW: 311.332
  • Catalog: Others
  • Density: 1.3±0.1 g/cm3
  • Boiling Point: 544.1±33.0 °C at 760 mmHg
  • Melting Point: 151-155 °C
  • Flash Point: 282.9±25.4 °C

Ozanezumab

Ozanezumab (GSK1223249) is an anti-Nogo-A (neurite outgrowth inhibitor A) monoclonal antibody. Ozanezumab can be used in amyotrophic lateral sclerosis (ALS) and multiple sclerosis research[1].

  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Glucosylsphingosine-d7

Glucosylsphingosine-d7 is deuterium labeled Glucosylsphingosine.

  • CAS Number: 2315262-29-2
  • MF: C24H40D7NO7
  • MW: 468.68
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

UCPH-102

UCPH-102 is a highly selective EAAT1 inhibitor with an IC50 of 0.43 µM. UCPH-102 exhibits a specific anti-proliferative effect on T-ALL cells. UCPH-102 also shows good blood-brain permeability, which can be used in studies of amyotrophic lateral sclerosis, Alzheimer’s disease, chronic pain and obsessive compulsive disorder[1][2][3][4].

  • CAS Number: 1229591-56-3
  • MF: C21H18N2O2
  • MW: 330.380
  • Catalog: Cancer
  • Density: 1.3±0.1 g/cm3
  • Boiling Point: 610.7±55.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 323.2±31.5 °C

H-Ser-Leu-Ser-Leu-Ser-Pro-Gly-OH trifluoroacetate salt

SLSLSPG can be obtained from the C-end of the heavy chain of human Igγ-1. SLSLSPG is a common variant in IgG[1].

  • CAS Number: 943235-75-4
  • MF: C28H49N7O11
  • MW: 659.73
  • Catalog: Others
  • Density: 1.3±0.1 g/cm3
  • Boiling Point: 1172.5±65.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 662.9±34.3 °C

BOC-3-IODO-D-ALANINE BENZYL ESTER

Boc-β-iodo-D-Ala-OBzl is an alanine derivative[1].

  • CAS Number: 125942-79-2
  • MF: C15H20INO4
  • MW: 405.22800
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: 80-84ºC(lit.)
  • Flash Point: N/A

elpamotide

Elpamotide is an epitope peptide derived from VEGFR2. Elpamotide induces cytotoxic T lymphocytes (CTLs) to kill VEGFR2-expressing endothelial cells. Elpamotide has potential immunostimulatory and antineoplastic activities. Elpamotide can be used in the research of cancer, such as pancreatic cancer[1][2].

  • CAS Number: 673478-49-4
  • MF: C47H76N16O13
  • MW: 1073.206
  • Catalog: Cancer
  • Density: 1.5±0.1 g/cm3
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Desmethylsildenafil-d8 citrate

Desmethylsildenafil-d8 (citrate) is the deuterium labeled Desmethylsildenafil citrate[1].

  • CAS Number: 1215071-06-9
  • MF: C27H28D8N6O11S
  • MW: 660.72300
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

2,5-Di-(tert-butyl)-4-methoxyphenol-3,6-d20

2,5-Di-(tert-butyl)-4-methoxyphenol-3,6-d20 is the deuterium labeled 2,5-Di-tert-butyl-4-methoxyphenol[1].

  • CAS Number: 1219802-07-9
  • MF: C15H24O2
  • MW: 236.350
  • Catalog: Others
  • Density: 1.0±0.1 g/cm3
  • Boiling Point: 337.8±42.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 129.2±12.8 °C

Cixutumumab

Cixutumumab (IMC-A12) is a humanized anti-IGF-1R monoclonal antibody with high affinity that inhibits ligand-dependent receptor activation and downstream signaling. Cixutumumab also mediates the internalization and degradation of IGF-IR. Cixutumumab shows broad-spectrum anti-tumour activity and can be used in studies of cancers such as lung cancer, malignancies, leukaemia, non-small cell lung cancer and prostate cancer[1].

  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

4-Methylumbelliferyl β-D-galactoside

4-Methylumbelliferyl β-D-galactopyranoside is a fluorescent substrate for β-galactosidase which, when cleaved, produces a water-soluble blue fluorescent coumarin fluorophore that can be detected using a fluoroenzymeter or fluorometer[1].

  • CAS Number: 6160-78-7
  • MF: C16H18O8
  • MW: 338.309
  • Catalog: Others
  • Density: 1.5±0.1 g/cm3
  • Boiling Point: 626.9±55.0 °C at 760 mmHg
  • Melting Point: 258-263ºC (dec.)
  • Flash Point: 233.9±25.0 °C

4-Methyl-5,6,7,8-tetrahydroquinoline

4-Methyl-5,6,7,8-tetrahydroquinoline, a tetrahydroquinoline alkaloid, is isolated from the roots of Glycyrrhiza uralensis Fisch[1].

  • CAS Number: 28971-03-1
  • MF: C10H13N
  • MW: 147.21700
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

1-Deoxynojirimycin

1-Deoxynojirimycin (DNJ, Duvoglustat) is a potent α-glucosidase inhibitor, suppresses postprandial blood glucose, thereby possibly preventing diabetes mellitus. Target: α-glucosidase1-Deoxynojirimycin is an alpha-glucosidase inhibitor, most commonly found in mulberry leaves. Although it can be obtained in small quantities by brewing an herbal tea from mulberry leaves, interest in commercial production has led to research on developing mulberry tea higher in DNJ, and on alternate routes of production, such as via Bacillusspecies.

  • CAS Number: 19130-96-2
  • MF: C6H13NO4
  • MW: 163.172
  • Catalog: Metabolic Disease
  • Density: 1.5±0.1 g/cm3
  • Boiling Point: 361.1±42.0 °C at 760 mmHg
  • Melting Point: 195-196°C
  • Flash Point: 197.3±18.5 °C

1-Methoxy-1H-indole-3-carboxylic acid

1-Methoxyindole-3-carboxylic acid (compound 5) is synthetic from a phytoalexin nucleophilic substitution reaction selectively at the 2-position[1].

  • CAS Number: 91913-76-7
  • MF: C10H9NO3
  • MW: 191.183
  • Catalog: Others
  • Density: 1.3±0.1 g/cm3
  • Boiling Point: 382.0±34.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 184.8±25.7 °C

Choline-d13 sulfate

Choline-d13 (sulfate) is the deuterium labeled Choline sulfate[1].

  • CAS Number: 2483831-84-9
  • MF: C5D13NO4S
  • MW: 196.31
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Lavandoside

Lavandoside is an active compound found from Lavandula spica flowers[1].

  • CAS Number: 117405-51-3
  • MF: C16H20O9
  • MW: 356.325
  • Catalog: Others
  • Density: 1.5±0.0 g/cm3
  • Boiling Point: 642.0±0.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 235.8±0.0 °C

H-D-Cys-OH.H2O.HCl

D-Cysteine hydrochloride is a cysteine derivative[1].

  • CAS Number: 32443-99-5
  • MF: C3H8ClNO2S
  • MW: 157.619
  • Catalog: Others
  • Density: N/A
  • Boiling Point: 293.9ºC at 760 mmHg
  • Melting Point: ~185 °C (dec.)
  • Flash Point: 131.5ºC

Cimiside B

Cimiside B, a glycoside alkaloid, isolated from the rhizome of Cimicifuga dahurica.

  • CAS Number: 152685-91-1
  • MF: C40H64O13
  • MW: 752.928
  • Catalog: Others
  • Density: 1.4±0.1 g/cm3
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Hydrazine sulfate-15N2

Hydrazine sulfate-15N2 is the 15N labeled Hydrazine sulfate[1].

  • CAS Number: 88491-70-7
  • MF: H6N2O4S
  • MW: 132.11000
  • Catalog: Others
  • Density: 1.391 g/mL at 25ºC
  • Boiling Point: 330ºC at 760 mmHg
  • Melting Point: 254ºC(lit.)
  • Flash Point: N/A

N3Ac-OPhOMe

N3Ac-OPhOMe is a click chemistry reagent containing an azide group. N3Ac-OPhOMe can be used for the research of various biochemical[1].

  • CAS Number: 2546513-31-7
  • MF: C9H9N3O3
  • MW: 207.19
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Fmoc-L-Cycpentala-OH

Fmoc-Cpa-OH is a compound containing both an amino group and a carboxyl group.

  • CAS Number: 371770-32-0
  • MF: C23H25NO4
  • MW: 379.449
  • Catalog: Others
  • Density: 1.2±0.1 g/cm3
  • Boiling Point: 598.0±33.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 315.4±25.4 °C

Fmoc-Glu(ODmab)-OH

Fmoc-Glu(ODmab)-OH is a glutamic acid derivative[1].

  • CAS Number: 268730-86-5
  • MF: C40H44N2O8
  • MW: 680.786
  • Catalog: Others
  • Density: 1.3±0.1 g/cm3
  • Boiling Point: 851.2±65.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 468.6±34.3 °C

Oxi 4503

Combretastatin A1 phosphate (Oxi4503; CA1P; Combretastatin A1 diphosphate) is a potent vascular disruptive agent. Combretastatin A1 phosphate exerts anti-angiogenic effects on tumors. Combretastatin A1 phosphate has the potential for the research of pancreatic neuroendocrine tumors[1][2].

  • CAS Number: 288847-35-8
  • MF: C18H22O12P2
  • MW: 492.30800
  • Catalog: Cancer
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Uvaol diacetate

Uvaol diacetate (Compound 5) is a type of triterpenoids derived from Nerium oleunder L. leaves [1].

  • CAS Number: 157000-65-2
  • MF: C34H54O4
  • MW: 526.79
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Mca-Pro-Leu-Gly-Leu-Glu-Glu-Ala-Dap(Dnp)-NH2 trifluoroacetate salt

Mca-Pro-Leu-Gly-Leu-Glu-Glu-Ala-Dap(Dnp)-NH2 is highly selective substrate for matrix metalloproteases 12 (MMP12) substrate with a kcat/Km value of 1.85*105 M-1s-1, and poor substrate of other MMPs with the exception of MMP13 (kcat/Km = 0.53*105 M-1s-1) and MMP9 (0.33*105 M-1s-1)[1].

  • CAS Number: 891198-38-2
  • MF: C53H70N12O20
  • MW: 1195.19000
  • Catalog: Cancer
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

kaempferoltetraacetate

Kaempferol tetraacetate (AF33) is a natural product. Kaempferol tetraacetate shows cytotoxicity[1][2].

  • CAS Number: 16274-11-6
  • MF: C23H18O10
  • MW: 454.383
  • Catalog: Cancer
  • Density: 1.4±0.1 g/cm3
  • Boiling Point: 609.7±55.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 263.9±31.5 °C