Chemsrc provides Others's classification. They are divided into Androgen Receptor, Aromatase, Estrogen Receptor/ERR, Progesterone Receptor, Thyroid Hormone Receptor, Others according to their Biological activity.


Anti-infection >
Arenavirus Bacterial CMV Enterovirus Filovirus Fungal HBV HCV HIV HSV Influenza Virus Parasite Reverse Transcriptase RSV SARS-CoV
Antibody-drug Conjugate >
ADC Cytotoxin ADC Linker Drug-Linker Conjugates for ADC PROTAC-linker Conjugate for PAC
Apoptosis >
Apoptosis Bcl-2 Family c-Myc Caspase DAPK Ferroptosis IAP MDM-2/p53 PKD RIP kinase Survivin Thymidylate Synthase TNF Receptor
Autophagy >
Autophagy LRRK2 ULK Mitophagy
Cell Cycle/DNA Damage >
Antifolate APC ATM/ATR Aurora Kinase Casein Kinase CDK Checkpoint Kinase (Chk) CRISPR/Cas9 Deubiquitinase DNA Alkylator/Crosslinker DNA-PK DNA/RNA Synthesis Eukaryotic Initiation Factor (eIF) G-quadruplex Haspin Kinase HDAC HSP IRE1 Kinesin LIM Kinase (LIMK) Microtubule/Tubulin Mps1 Nucleoside Antimetabolite/Analog p97 PAK PARP PERK Polo-like Kinase (PLK) PPAR RAD51 ROCK Sirtuin SRPK Telomerase TOPK Topoisomerase Wee1
Cytoskeleton >
Arp2/3 Complex Dynamin Gap Junction Protein Integrin Kinesin Microtubule/Tubulin Mps1 Myosin PAK
Epigenetics >
AMPK Aurora Kinase DNA Methyltransferase Epigenetic Reader Domain HDAC Histone Acetyltransferase Histone Demethylase Histone Methyltransferase JAK MicroRNA PARP PKC Sirtuin Protein Arginine Deiminase
GPCR/G Protein >
5-HT Receptor Adenosine Receptor Adenylate Cyclase Adiponectin Receptor Adrenergic Receptor Angiotensin Receptor Bombesin Receptor Bradykinin Receptor Cannabinoid Receptor CaSR CCR CGRP Receptor Cholecystokinin Receptor CRFR CXCR Dopamine Receptor EBI2/GPR183 Endothelin Receptor GHSR Glucagon Receptor Glucocorticoid Receptor GNRH Receptor GPCR19 GPR109A GPR119 GPR120 GPR139 GPR40 GPR55 GPR84 Guanylate Cyclase Histamine Receptor Imidazoline Receptor Leukotriene Receptor LPL Receptor mAChR MCHR1 (GPR24) Melatonin Receptor mGluR Motilin Receptor Neurokinin Receptor Neuropeptide Y Receptor Neurotensin Receptor Opioid Receptor Orexin Receptor (OX Receptor) Oxytocin Receptor P2Y Receptor Prostaglandin Receptor Protease-Activated Receptor (PAR) Ras RGS Protein Sigma Receptor Somatostatin Receptor TSH Receptor Urotensin Receptor Vasopressin Receptor Melanocortin Receptor
Immunology/Inflammation >
Aryl Hydrocarbon Receptor CCR Complement System COX CXCR FLAP Histamine Receptor IFNAR Interleukin Related IRAK MyD88 NO Synthase NOD-like Receptor (NLR) PD-1/PD-L1 PGE synthase Salt-inducible Kinase (SIK) SPHK STING Thrombopoietin Receptor Toll-like Receptor (TLR) Arginase
JAK/STAT Signaling >
EGFR JAK Pim STAT
MAPK/ERK Pathway >
ERK JNK KLF MAP3K MAP4K MAPKAPK2 (MK2) MEK Mixed Lineage Kinase MNK p38 MAPK Raf Ribosomal S6 Kinase (RSK)
Membrane Transporter/Ion Channel >
ATP Synthase BCRP Calcium Channel CFTR Chloride Channel CRAC Channel CRM1 EAAT2 GABA Receptor GlyT HCN Channel iGluR Monoamine Transporter Monocarboxylate Transporter Na+/Ca2+ Exchanger Na+/HCO3- Cotransporter Na+/K+ ATPase nAChR NKCC P-glycoprotein P2X Receptor Potassium Channel Proton Pump SGLT Sodium Channel TRP Channel URAT1
Metabolic Enzyme/Protease >
15-PGDH 5 alpha Reductase 5-Lipoxygenase Acetyl-CoA Carboxylase Acyltransferase Adenosine Deaminase Adenosine Kinase Aldehyde Dehydrogenase (ALDH) Aldose Reductase Aminopeptidase Angiotensin-converting Enzyme (ACE) ATGL ATP Citrate Lyase Carbonic Anhydrase Carboxypeptidase Cathepsin CETP COMT Cytochrome P450 Dipeptidyl Peptidase Dopamine β-hydroxylase E1/E2/E3 Enzyme Elastase Enolase FAAH FABP Factor Xa Farnesyl Transferase Fatty Acid Synthase (FAS) FXR Glucokinase GSNOR Gutathione S-transferase HCV Protease Hexokinase HIF/HIF Prolyl-Hydroxylase HIV Integrase HIV Protease HMG-CoA Reductase (HMGCR) HSP Indoleamine 2,3-Dioxygenase (IDO) Isocitrate Dehydrogenase (IDH) Lactate Dehydrogenase LXR MAGL Mineralocorticoid Receptor Mitochondrial Metabolism MMP Nampt NEDD8-activating Enzyme Neprilysin PAI-1 PDHK PGC-1α Phosphatase Phosphodiesterase (PDE) Phospholipase Procollagen C Proteinase Proteasome Pyruvate Kinase RAR/RXR Renin ROR Ser/Thr Protease SGK Stearoyl-CoA Desaturase (SCD) Thrombin Tryptophan Hydroxylase Tyrosinase Xanthine Oxidase
Neuronal Signaling >
5-HT Receptor AChE Adenosine Kinase Amyloid-β Beta-secretase CaMK CGRP Receptor COMT Dopamine Receptor Dopamine Transporter FAAH GABA Receptor GlyT iGluR Imidazoline Receptor mAChR Melatonin Receptor Monoamine Oxidase nAChR Neurokinin Receptor Opioid Receptor Serotonin Transporter γ-secretase
NF-κB >
NF-κB IKK Keap1-Nrf2 MALT1
PI3K/Akt/mTOR >
Akt AMPK ATM/ATR DNA-PK GSK-3 MELK mTOR PDK-1 PI3K PI4K PIKfyve PTEN
PROTAC >
PROTAC E3 Ligase Ligand-Linker Conjugate Ligand for E3 Ligase PROTAC Linker PROTAC-linker Conjugate for PAC
Protein Tyrosine Kinase/RTK >
Ack1 ALK Bcr-Abl BMX Kinase Btk c-Fms c-Kit c-Met/HGFR Discoidin Domain Receptor DYRK EGFR Ephrin Receptor FAK FGFR FLT3 IGF-1R Insulin Receptor IRAK Itk PDGFR PKA Pyk2 ROS Src Syk TAM Receptor Trk Receptor VEGFR
Stem Cell/Wnt >
Casein Kinase ERK Gli GSK-3 Hedgehog Hippo (MST) JAK Notch Oct3/4 PKA Porcupine ROCK sFRP-1 Smo STAT TGF-beta/Smad Wnt YAP β-catenin γ-secretase
TGF-beta/Smad >
TGF-beta/Smad PKC ROCK TGF-β Receptor
Vitamin D Related >
VD/VDR
Others >
Androgen Receptor Aromatase Estrogen Receptor/ERR Progesterone Receptor Thyroid Hormone Receptor Others

Zinc dihexonate

Zinc Gluconate has the potential for the research of common cold, cancer, and a nutrition supplement as a food additive[1].

  • CAS Number: 4468-02-4
  • MF: C12H22O14Zn
  • MW: 455.704
  • Catalog: Others
  • Density: N/A
  • Boiling Point: 673.6ºC at 760 mmHg
  • Melting Point: 131ºC
  • Flash Point: 375.2ºC

Amino Albendazole

ABZ-amine (Amino albendazole) is an impurity of Albendazole. Albendazole is a member of the benzimidazole compounds used as a drug indicated for the treatment of a variety of worm infestations[1][2].

  • CAS Number: 80983-36-4
  • MF: C10H13N3S
  • MW: 207.29500
  • Catalog: Others
  • Density: 1.26g/cm3
  • Boiling Point: 438.6ºC at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 219ºC

TAMRA hydrazide (6-isomer)

TAMRA hydrazide (6-isomer) is a click chemistry reagent that can be coupled to carbonyl compounds. The dye hydrazide in TAMRA hydrazide (6-isomer) labels carbonyl compounds such as aldehydes and ketones. TAMRA in TAMRA hydrazide (6-isomer) is a xanthene red fluorophore that reacts with terminal alkynes.

  • CAS Number: 2183440-67-5
  • MF: C25H25ClN4O4
  • MW: 480.94
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Acetyl-Hirudin (54-65) (sulfated)

Acetyl-Hirudin (54-65) (sulfated) binds directly to thrombin-rHCII(L444R) and disrupts interactions between the N-terminal acidic domain of rHCII and anion-binding exosite I of thrombin that serves to stabilize the complex[1].

  • CAS Number: 125441-00-1
  • MF: C68H95N13O29S
  • MW: 1590.617
  • Catalog: Metabolic Disease
  • Density: 1.4±0.1 g/cm3
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

NF(N-Me)GA(N-Me)IL

NF(N-Me)GA(N-Me)IL is a biological active peptide. (This amino acids 22 to 27 fragment is a modification of the human islet amyloid polypeptide hIAPP (NFGAIL) with N-methylation of the amide bonds at G24 and I26. The introduction of two N-methyl rests in the amyloid-core-containing sequence NFGAIL converts this amyloidogenic and cytotoxic sequence into non-amyloidogenic and non-cytotoxic peptide. The peptide is able to bind with high-affinity full-length hIAPP and to inhibit its fibrillogenesis.)

  • CAS Number: 409085-42-3
  • MF: C32H51N7O8
  • MW: 661.79
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Ecteinascidin-Analog-1

Ecteinascidin-Analog-1 is a useful intermediate for chemical sythesis of Ecteinascidin analogues; Ecteinascidins is a family of tetrahydroisoquinoline alkaloids with wide range of antitumor and antimicrobial activities.

  • CAS Number: 874758-58-4
  • MF: C31H44N2O9
  • MW: 588.68900
  • Catalog: Cancer
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Schnurri-3 inhibitor-1

Schnurri-3 inhibitor-1 is a potent schnurri-3 inhibitor which is an essential regulator of adult bone formation. Schnurri-3 inhibitor-1 can inhibit Shn3 with EF1alpha promoter in osteoblast cell line Shn3FFL with an AC50 value of 2.09 μM. Schnurri-3 inhibitor-1 can be used to research osteoporosis[1].

  • CAS Number: 736154-60-2
  • MF: C12H10F2N2O2S
  • MW: 284.28
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Limocitrin-3-rutinoside

Limocitrin-3-rutinoside is a member of flavonoids and a glycoside. Limocitrin-3-rutinoside can be isolated from peach fruit[1].

  • CAS Number: 79384-27-3
  • MF: C29H34O17
  • MW: 654.57
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Kinesore

Kinesore is an inhibitor of the KLC2-SKIP Interaction.

  • CAS Number: 363571-83-9
  • MF: C20H16Br2N4O4
  • MW: 536.173
  • Catalog: Others
  • Density: 1.7±0.1 g/cm3
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

N-Boc-phenyl-alaninal-d5

N-Boc-phenyl-alaninal-d5 is the deuterium labeled Aminoisobutyric acid hydrochloride[1].

  • CAS Number: 1217724-86-1
  • MF: C14H14D5NO3
  • MW: 254.34
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

1,2-Dipalmitoyl-sn-glycero-O-ethyl-3-phosphoryl choline chloride

16:0 EPC chloride, a P-O-ethyl derivative, is a saturated cationic lipid. 16:0 EPC chloride can serve as a DNA and RNA transfecting agent. 16:0 EPC chloride can be used as a co-adjuvant for preparing vaccines and promote drug delivery[1].

  • CAS Number: 328250-18-6
  • MF: C42H85ClNO8P
  • MW: 798.553
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

L-6424

L-6424 inhibits T3 binding to α1-T3R and β1-T3R[1].

  • CAS Number: 147030-50-0
  • MF: C19H17IO3
  • MW: 420.24100
  • Catalog: Metabolic Disease
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Azure A

Giemsa stain can stain chromatin and nuclear membrane. Giemsa stain histopathologic detection of malaria and other microorganisms, such as Histoplasma, LeishmaniaToxoplasma, and Pneumocystis .Giemsa stain can used be in histology and microbiology[1].

  • CAS Number: 51811-82-6
  • MF: C14H14ClN3S
  • MW: 291.799
  • Catalog: Others
  • Density: 0.99
  • Boiling Point: 543ºC at 760mmHg
  • Melting Point: 300 °C(lit.)
  • Flash Point: 15 °C

3,5-Dihydroxyphenyl β-D-glucopyranoside

Phlorin (Phloroglucinol β-D-glucoside) is a phloroglucinol (PG) glucoside[1].

  • CAS Number: 28217-60-9
  • MF: C12H16O8
  • MW: 288.251
  • Catalog: Others
  • Density: 1.7±0.1 g/cm3
  • Boiling Point: 598.8±50.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 315.9±30.1 °C

Hypoglycemic agent 1

Hypoglycemic agent 1 acts as a therapeutic and/or prophylactic agent for diabetes. Hypoglycemic agent 1 has an action for lowering blood sugar[1].

  • CAS Number: 2253733-57-0
  • MF: C25H24FN5O4
  • MW: 477.49
  • Catalog: Metabolic Disease
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Gastric mucin

Gastric mucin is a large glycoprotein which is thought to play a major role in the protection of the gastrointestinal tract from acid, proteases, pathogenic microorganisms, and mechanical trauma.

  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

2: PN: US20040072744 SEQID: 2 claimed protein

2: PN: US20040072744 SEQID: 2 claimed protein is a synthetic peptide, used for the research of Down's syndrome and schizophrenia.

  • CAS Number: 389572-87-6
  • MF: C43H67N13O17S
  • MW: 1070.13
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Sulfo-Cy5-tetrazine

Cy5 Tetrazine is a water-soluble, pH-insensitive from pH 4 to pH 10, far-red-fluorescent probe with excitation ideally suited for the 633 nm or 647 nm laser lines. Its absorption and emission spactra are almost identical to those of Alexa Fluor 647, CF 647 Dye, or any other Cyanine5 based fluorescent dyes.

  • CAS Number: 1801695-57-7
  • MF: C43H49N7O10S3
  • MW: 920.09
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

4-Methylcaprylic acid

4-Methyloctanoic acid is a natural compound mainly responsible for the characteristic goaty sheepy flavour of sheep and goat milk[1].

  • CAS Number: 54947-74-9
  • MF: C9H18O2
  • MW: 158.238
  • Catalog: Others
  • Density: 0.9±0.1 g/cm3
  • Boiling Point: 253.4±8.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 129.7±6.9 °C

H-Leu-Ser-Phe-OH

H-Leu-Ser-Phe-OH is a biologically active peptide.

  • CAS Number: 40290-77-5
  • MF: C18H27N3O5
  • MW: 365.424
  • Catalog: Others
  • Density: 1.2±0.1 g/cm3
  • Boiling Point: 691.2±55.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 371.8±31.5 °C

S186

S186 is a kind of sodium salts of calcium-acetylpropylamine phosphonate(APA); a new strontium-specific chelating agent.IC50 value:Target: In a case test for 4 person who took 90Sr in due to an internal contaminated accident, the APAP was adminstrated intramuscularly once a day for 3 days, the increase excretion of 90Sr was obvious and no side effects was observed among them. Recently, S186 has also been approved by Shanghai Municipal Health Bureau for emergency medical use in China.

  • CAS Number: 97759-16-5
  • MF: C5H13CaNNaO7P2
  • MW: 324.17500
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

BI 6015

BI-6015 is a hepatocyte nuclear factor 4α (HNF4α) antagonist that can inhibit the expression of known HNF4α target genes. BI6015 represses insulin promoter activity through HNF4α antagonism. BI-6015 can be used for the research of cancer and diabetes[1].

  • CAS Number: 93987-29-2
  • MF: C15H13N3O4S
  • MW: 331.35
  • Catalog: Cancer
  • Density: 1.5±0.1 g/cm3
  • Boiling Point: 570.6±60.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 298.9±32.9 °C

Germacrene D

(Rac)-Germacrene D is a racemate of Germacrene D. Germacrene D has antibacterial and antifungal activities and can be used as an adjuvant agent in the application of aminoglycosides and azoles[1].

  • CAS Number: 37839-63-7
  • MF: C15H24
  • MW: 204.35
  • Catalog: Others
  • Density: 0.85g/cm3
  • Boiling Point: 279.7ºC at 760mmHg
  • Melting Point: N/A
  • Flash Point: 111.9ºC

Dansyl Ethylenediamine

Dansyl ethylenediamine is a fluorescent probe. Dansyl ethylenediamine can be used for synthesis of protein-imprinted polymers which is capable of specific transduction of protein binding events into fluorescent signal change[1].

  • CAS Number: 35060-08-3
  • MF: C14H19N3O2S
  • MW: 293.38500
  • Catalog: Others
  • Density: 1.262g/cm3
  • Boiling Point: 470.2ºC at 760mmHg
  • Melting Point: 145-146ºC
  • Flash Point: 238.1ºC

Acetylatractylodinol

Acetylatractylodinol, isolated from Atractylodes lancea, possesses antioxidant activity[1].

  • CAS Number: 61582-39-6
  • MF: C15H14O4
  • MW: 258.26900
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

5,9-Dihydroxy-8-methoxy-2,2-dimethyl-7-(3-methyl-2-buten-1-yl)-3,4-dihydro-2H,6H-pyrano[3,2-b]xanthen-6-one

3-Isomangostin, extracted from Garciniamangostana.L. shell, is a potent MutT homologue 1 (MTH1) inhibitor with an IC50 value of 52 nM. 3-isomangostin would be an attractive chemical tool for the development of anticancer agents[1].

  • CAS Number: 19275-46-8
  • MF: C24H26O6
  • MW: 410.460
  • Catalog: Cancer
  • Density: 1.3±0.1 g/cm3
  • Boiling Point: 615.9±55.0 °C at 760 mmHg
  • Melting Point: 155-160ºC
  • Flash Point: 212.3±25.0 °C

3-Methylphenol acetate

m-Tolyl acetate is a intermediate of organic synthesis.

  • CAS Number: 122-46-3
  • MF: C9H10O2
  • MW: 150.17400
  • Catalog: Others
  • Density: 1.04 g/mL at 25 °C(lit.)
  • Boiling Point: 210-213 °C(lit.)
  • Melting Point: N/A
  • Flash Point: 203 °F

MARK-IN-1

MARK-IN-1 is a potent microtubule affinity regulating kinase (MARK) inhibitor with an IC50 of <0.25 nM.

  • CAS Number: 1109283-93-3
  • MF: C22H23F2N7OS
  • MW: 471.52600
  • Catalog: Neurological Disease
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

1,2-Distearoyl-sn-glycero-3-phosphorylcholine-d9

1,2-Distearoyl-sn-glycero-3-phosphorylcholine-d9 is deuterium labeled 1,2-Distearoyl-sn-glycero-3-phosphorylcholine. 1,2-Distearoyl-sn-glycero-3-phosphorylcholine (1,2-Distearoyl-sn-glycero-3-PC; DSPC) is a cylindrical-shaped lipid. 1,2-Distearoyl-sn-glyc

  • CAS Number: 326495-36-7
  • MF: C44H79D9NO8P
  • MW: 799.20
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

WAY-325811

WAY-325811 is an active molecule.

  • CAS Number: 869632-12-2
  • MF: C18H18N2O2S
  • MW: 326.41
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A