An antifungal agent is a drug that selectively eliminates fungal pathogens from a host with minimal toxicity to the host. Classes: 1. Polyene Antifungal Drugs: Amphotericin, nystatin, and pimaricin interact with sterols in the cell membrane (ergosterol in fungi, cholesterol in humans) to form channels through which small molecules leak from the inside of the fungal cell to the outside. 2. Azole Antifungal Drugs: Fluconazole, itraconazole, and ketoconazole inhibit cytochrome P450-dependent enzymes (particularly C14-demethylase) involved in the biosynthesis of ergosterol, which is required for fungal cell membrane structure and function. 3. Allylamine and Morpholine Antifungal Drugs: lylamines (naftifine, terbinafine) inhibit ergosterol biosynthesis at the level of squalene epoxidase. The morpholine drug, amorolfine, inhibits the same pathway at a later step. 4. Antimetabolite Antifungal Drugs: 5-Fluorocytosine acts as an inhibitor of both DNA and RNA synthesis via the intracytoplasmic conversion of 5-fluorocytosine to 5-fluorouracil.


Anti-infection >
Arenavirus Bacterial CMV Enterovirus Filovirus Fungal HBV HCV HIV HSV Influenza Virus Parasite Reverse Transcriptase RSV SARS-CoV
Antibody-drug Conjugate >
ADC Cytotoxin ADC Linker Drug-Linker Conjugates for ADC PROTAC-linker Conjugate for PAC
Apoptosis >
Apoptosis Bcl-2 Family c-Myc Caspase DAPK Ferroptosis IAP MDM-2/p53 PKD RIP kinase Survivin Thymidylate Synthase TNF Receptor
Autophagy >
Autophagy LRRK2 ULK Mitophagy
Cell Cycle/DNA Damage >
Antifolate APC ATM/ATR Aurora Kinase Casein Kinase CDK Checkpoint Kinase (Chk) CRISPR/Cas9 Deubiquitinase DNA Alkylator/Crosslinker DNA-PK DNA/RNA Synthesis Eukaryotic Initiation Factor (eIF) G-quadruplex Haspin Kinase HDAC HSP IRE1 Kinesin LIM Kinase (LIMK) Microtubule/Tubulin Mps1 Nucleoside Antimetabolite/Analog p97 PAK PARP PERK Polo-like Kinase (PLK) PPAR RAD51 ROCK Sirtuin SRPK Telomerase TOPK Topoisomerase Wee1
Cytoskeleton >
Arp2/3 Complex Dynamin Gap Junction Protein Integrin Kinesin Microtubule/Tubulin Mps1 Myosin PAK
Epigenetics >
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GPCR/G Protein >
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Immunology/Inflammation >
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JAK/STAT Signaling >
EGFR JAK Pim STAT
MAPK/ERK Pathway >
ERK JNK KLF MAP3K MAP4K MAPKAPK2 (MK2) MEK Mixed Lineage Kinase MNK p38 MAPK Raf Ribosomal S6 Kinase (RSK)
Membrane Transporter/Ion Channel >
ATP Synthase BCRP Calcium Channel CFTR Chloride Channel CRAC Channel CRM1 EAAT2 GABA Receptor GlyT HCN Channel iGluR Monoamine Transporter Monocarboxylate Transporter Na+/Ca2+ Exchanger Na+/HCO3- Cotransporter Na+/K+ ATPase nAChR NKCC P-glycoprotein P2X Receptor Potassium Channel Proton Pump SGLT Sodium Channel TRP Channel URAT1
Metabolic Enzyme/Protease >
15-PGDH 5 alpha Reductase 5-Lipoxygenase Acetyl-CoA Carboxylase Acyltransferase Adenosine Deaminase Adenosine Kinase Aldehyde Dehydrogenase (ALDH) Aldose Reductase Aminopeptidase Angiotensin-converting Enzyme (ACE) ATGL ATP Citrate Lyase Carbonic Anhydrase Carboxypeptidase Cathepsin CETP COMT Cytochrome P450 Dipeptidyl Peptidase Dopamine β-hydroxylase E1/E2/E3 Enzyme Elastase Enolase FAAH FABP Factor Xa Farnesyl Transferase Fatty Acid Synthase (FAS) FXR Glucokinase GSNOR Gutathione S-transferase HCV Protease Hexokinase HIF/HIF Prolyl-Hydroxylase HIV Integrase HIV Protease HMG-CoA Reductase (HMGCR) HSP Indoleamine 2,3-Dioxygenase (IDO) Isocitrate Dehydrogenase (IDH) Lactate Dehydrogenase LXR MAGL Mineralocorticoid Receptor Mitochondrial Metabolism MMP Nampt NEDD8-activating Enzyme Neprilysin PAI-1 PDHK PGC-1α Phosphatase Phosphodiesterase (PDE) Phospholipase Procollagen C Proteinase Proteasome Pyruvate Kinase RAR/RXR Renin ROR Ser/Thr Protease SGK Stearoyl-CoA Desaturase (SCD) Thrombin Tryptophan Hydroxylase Tyrosinase Xanthine Oxidase
Neuronal Signaling >
5-HT Receptor AChE Adenosine Kinase Amyloid-β Beta-secretase CaMK CGRP Receptor COMT Dopamine Receptor Dopamine Transporter FAAH GABA Receptor GlyT iGluR Imidazoline Receptor mAChR Melatonin Receptor Monoamine Oxidase nAChR Neurokinin Receptor Opioid Receptor Serotonin Transporter γ-secretase
NF-κB >
NF-κB IKK Keap1-Nrf2 MALT1
PI3K/Akt/mTOR >
Akt AMPK ATM/ATR DNA-PK GSK-3 MELK mTOR PDK-1 PI3K PI4K PIKfyve PTEN
PROTAC >
PROTAC E3 Ligase Ligand-Linker Conjugate Ligand for E3 Ligase PROTAC Linker PROTAC-linker Conjugate for PAC
Protein Tyrosine Kinase/RTK >
Ack1 ALK Bcr-Abl BMX Kinase Btk c-Fms c-Kit c-Met/HGFR Discoidin Domain Receptor DYRK EGFR Ephrin Receptor FAK FGFR FLT3 IGF-1R Insulin Receptor IRAK Itk PDGFR PKA Pyk2 ROS Src Syk TAM Receptor Trk Receptor VEGFR
Stem Cell/Wnt >
Casein Kinase ERK Gli GSK-3 Hedgehog Hippo (MST) JAK Notch Oct3/4 PKA Porcupine ROCK sFRP-1 Smo STAT TGF-beta/Smad Wnt YAP β-catenin γ-secretase
TGF-beta/Smad >
TGF-beta/Smad PKC ROCK TGF-β Receptor
Vitamin D Related >
VD/VDR
Others >
Androgen Receptor Aromatase Estrogen Receptor/ERR Progesterone Receptor Thyroid Hormone Receptor Others

Dihydroaltenuene B

Dihydroaltenuene B is a potent mushroom tyrosinase inhibitor with an IC50 of 38.33 µM. Dihydroaltenuene B shows the hydrogen bonding interactions between the 3-OH and 4’-OH and the His244, Met280 and Gly281 residues of tyrosinase[1].

  • CAS Number: 887751-89-5
  • MF: C15H18O6
  • MW: 294.30
  • Catalog: Fungal
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Tetrahydrojatrorrhizine

Corypalmine is an alkaloid from Corydalis chaerophylla. Corypalmine is an antifungal.

  • CAS Number: 27313-86-6
  • MF: C20H23NO4
  • MW: 341.40100
  • Catalog: Fungal
  • Density: 1.29g/cm3
  • Boiling Point: 501.2ºC at 760mmHg
  • Melting Point: N/A
  • Flash Point: 256.9ºC

Antifungal agent 31

Antifungal agent 31 (compound 12) is a potent and orally active triazole antifungal agents with a pyrrolotriazinone scaffold. Antifungal agent 31 shows antifungal activity against Candida spp. and filamentous fungi. Antifungal agent 31 significantly reduced mortality rates and kidney fungal burden in two murine models of lethal systemic infections[1].

  • CAS Number: 2077083-94-2
  • MF: C25H22F2N6O3
  • MW: 492.48
  • Catalog: Fungal
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

JUSTICIDIN B

Justicidin B is a potent anticancer lignan and proapoptotic agent. Justicidin B is also a bone resorption inhibitor, and has strong antiviral, fungicidal, antiprotozoal effects. Justicidin B significantly inhibits platelet aggregation[1][2][3].

  • CAS Number: 17951-19-8
  • MF: C21H16O6
  • MW: 364.34800
  • Catalog: Fungal
  • Density: 1.376g/cm3
  • Boiling Point: 601.9ºC at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 266ºC

(+)-Piresil diacetate

(+)-Pinoresinol diacetate is an antifungal agent that can be isolated from Sambucus williamsii[1].

  • CAS Number: 32971-25-8
  • MF: C24H26O8
  • MW: 442.458
  • Catalog: Fungal
  • Density: 1.2±0.1 g/cm3
  • Boiling Point: 539.9±50.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 232.4±30.2 °C

Aliconazole

Aliconazole is an antifungal imidazole derivative.

  • CAS Number: 63824-12-4
  • MF: C18H13Cl3N2
  • MW: 363.66800
  • Catalog: Fungal
  • Density: 1.29g/cm3
  • Boiling Point: 545ºC at 760mmHg
  • Melting Point: N/A
  • Flash Point: 283.4ºC

Pseudolaric Acid A

Pseudolaric Acid A is a diterpene acid isolated from Pseudolarix kaempferi, has antifungal, cytotoxic and antifertile activities[1][2][3].

  • CAS Number: 82508-32-5
  • MF: C22H28O6
  • MW: 388.454
  • Catalog: Fungal
  • Density: 1.23
  • Boiling Point: 571.5±50.0 °C at 760 mmHg
  • Melting Point: 206-207 ºC
  • Flash Point: 196.6±23.6 °C

TMV-IN-5

TMV-IN-5 (compound 1a) is an anti-plant virus/fungal agent. TMV-IN-5 inhibits viral assembly by binding to tobacco mosaic virus (TMV) CP. TMV-IN-5 can be used in the development of pesticides[1].

  • CAS Number: 1207318-92-0
  • MF: C22H23N3S
  • MW: 361.50
  • Catalog: Fungal
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Fenpropidin

Fenpropidin is a sterol biosynthesis inhibitor fungicide[1].

  • CAS Number: 67306-00-7
  • MF: C19H31N
  • MW: 273.45600
  • Catalog: Fungal
  • Density: 0.924 g/cm3
  • Boiling Point: 368.9ºC at 760 mmHg
  • Melting Point: 25°C
  • Flash Point: 159.3ºC

4,9-Dihydroxy-α-lapachone

Catalpanp-1 is a potent anti-microbial agent. Catalpanp-1 has strong antimicrobial effect on yeast, bacteria, fungi and the like[1].

  • CAS Number: 56473-67-7
  • MF: C15H14O5
  • MW: 274.27
  • Catalog: Bacterial
  • Density: 1.5±0.1 g/cm3
  • Boiling Point: 495.3±45.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 190.0±22.2 °C

Oligomycin

Oligomycins are macrolides created by Streptomyces species that can be toxic to other organisms through their ability to inhibit mitochondrial membrane-bound ATP synthases. The mitochondrial F1FO ATP synthase can switch to an ATP hydrolase during ischemia, so that, under these conditions, inhibition by oligomycins will reduce ATP depletion rather than block ATP synthesis.

  • CAS Number: 1404-19-9
  • MF: C135H220O33
  • MW: 2371.171
  • Catalog: Fungal
  • Density: 1.14 g/cm3
  • Boiling Point: 886.3ºC at 760 mmHg
  • Melting Point: 84-100ºC
  • Flash Point: 252ºC

5-epi-Jinkoheremol

5-epi-Jinkoheremol exhibits more potent fungicidal activity than validamycin.

  • CAS Number: 2567930-96-3
  • MF: C15H26O
  • MW: 222.37
  • Catalog: Fungal
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Tolnaftate-d7

Tolnaftate D7 (NP-27 D7) is the deuterium labeled Tolnaftate. Tolnaftate (NP-27) is a synthetic thiocarbamate used as an anti-fungal agent[1][2].

  • CAS Number: 1329835-64-4
  • MF: C19H10D7NOS
  • MW: 314.453
  • Catalog: Fungal
  • Density: 1.2±0.1 g/cm3
  • Boiling Point: 453.4±38.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 228.0±26.8 °C

Tolytoxin

Tolytoxin, a bioactive metabolite from cyanobacteria, is a potent antifungal antibiotic, exhibiting MICs of 0.25-8 nmol. Tolytoxin is a cyanobacterial macrolide that targets actin by inhibition of its polymerization. Tolytoxin has cytotoxic effects in cancer cells[1].

  • CAS Number: 127999-44-4
  • MF: C46H75NO13
  • MW: 850.09
  • Catalog: Fungal
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Anidulafungin

Anidulafungin is a new semisynthetic echinocandin with antifungal potency.

  • CAS Number: 166663-25-8
  • MF: C58H73N7O17
  • MW: 1140.237
  • Catalog: Fungal
  • Density: 1.5±0.1 g/cm3
  • Boiling Point: 1477.0±65.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 847.0±34.3 °C

Agoniadin

Plumieride is an antifungal agent. Plumieride has strong fungitoxicity against some dermatophytes. Plumieride has little cytotoxic activity against the P388 leukaemia cell line with an IC50 of 85 μg/mL[1].

  • CAS Number: 511-89-7
  • MF: C21H26O12
  • MW: 470.42
  • Catalog: Fungal
  • Density: 1.6±0.1 g/cm3
  • Boiling Point: 771.4±60.0 °C at 760 mmHg
  • Melting Point: 156-158°; mp 224-225°
  • Flash Point: 269.2±26.4 °C

Terbinafine

Terbinafine (TDT 067) is an antifungal medication used to treat fungal infections. It is a potent non-competitive inhibitor of squalene epoxidase from Candida with a Ki of 30 nM.

  • CAS Number: 91161-71-6
  • MF: C21H25N
  • MW: 291.430
  • Catalog: Fungal
  • Density: 1.0±0.1 g/cm3
  • Boiling Point: 417.9±33.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 183.7±22.3 °C

tribenuron-methyl [ANSI]

Tribenuron-methyl, a sulfonylurea herbicide agent, can be used as the fungicide agent. Tribenuron-methyl plays an important role in controlling the weeds and diseases in wheat field[1].

  • CAS Number: 101200-48-0
  • MF: C15H17N5O6S
  • MW: 395.39
  • Catalog: Fungal
  • Density: 1.4±0.1 g/cm3
  • Boiling Point: 376.6ºC
  • Melting Point: 141°C
  • Flash Point: 181.6ºC

Bikaverin

Bikaverin (Lycopersin) is a reddish pigment produced by different fungal species. Bikaverin shows antibiotic properties against certain protozoa and fungi[1].

  • CAS Number: 33390-21-5
  • MF: C20H14O8
  • MW: 382.32000
  • Catalog: Fungal
  • Density: 1.61g/cm3
  • Boiling Point: 719.8ºC at 760mmHg
  • Melting Point: N/A
  • Flash Point: 263.3ºC

1-Benzopyrylium,5,7-dihydroxy-2-(4-hydroxyphenyl)-, chloride (1:1)

Apigeninidin (Gesneridin) chloride, a 3‐deoxyanthocyanidin, is a fungal growth inhibitor. Apigeninidin chloride is a bioactive red biocolorant[1].

  • CAS Number: 1151-98-0
  • MF: C15H11ClO4
  • MW: 290.69800
  • Catalog: Fungal
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Fmoc-Gly-OH-1-13C

Fmoc-Gly-OH-1-13C is a 13C-labeled Carbendazim. Carbendazim is a potent and orally active broad-spectrum benzimidazole fungicide and can be acts as a pesticide for fungal diseases research, such as Seproria, Fusarium and Sclerotina[1][3]. Carbendazim is a

  • CAS Number: 197965-68-7
  • MF: C1613CH15NO4
  • MW: 298.30
  • Catalog: Fungal
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Cyclo(L-Phe-L-Val)

Cyclo(L-Phe-L-Val) is a potent inhibitor of enzymes isocitrate lyase (ICL) (IC50=27 μg/mL). cyclo(L-Phe-L-Val) inhibits the gene transcription of ICL in C. albicans under C2-carbon-utilizing conditions[1].

  • CAS Number: 35590-86-4
  • MF: C14H18N2O2
  • MW: 246.30
  • Catalog: Fungal
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

macrocarpal C

Macrocarpal C can be isolated from the 95 % ethanol extract of fresh leaves of E. globulus. Macrocarpal C inhibits the growth of T. mentagrophytes via an increase in the permeability of the fungal membrane. Macrocarpal C increases the production of intracellular ROS and? induces apoptosis as a consequence of DNA fragmentation[1].

  • CAS Number: 142628-53-3
  • MF: C28H38O5
  • MW: 454.60
  • Catalog: Fungal
  • Density: 1.2±0.1 g/cm3
  • Boiling Point: 503.9±50.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 272.6±26.6 °C

Sakuranetin

Sakuranetin is a rice flavonoid phytoalexin, shows strong antifungal activity[1]. Sakuranetin has anti-inflammatory and antioxidative activities. Sakuranetin ameliorates LPS-induced acute lung injury[2].

  • CAS Number: 2957-21-3
  • MF: C16H14O5
  • MW: 286.28
  • Catalog: Fungal
  • Density: 1.4±0.1 g/cm3
  • Boiling Point: 555.9±50.0 °C at 760 mmHg
  • Melting Point: 153-154ºC
  • Flash Point: 212.4±23.6 °C

Efungumab

Efungumab is a monoclonal antibody with antifungal activity. Efungumab binds to HSP 90, preventing a conformational change needed for fungal viability. Efungumab can be used for research on invasive candidiasis (IC)[1].

  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

SP-B peptide

SP-B peptide is an antimicrobial peptide. SP-B peptide has antifungal activity against strains of Cryptococcus neoformans, Candida albicans and Aspergillus fumigatus[1]

  • CAS Number: 865714-65-4
  • MF: C90H134N24O22
  • MW: 1904.17
  • Catalog: Fungal
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Magnoflorine

(+)-Magnoflorine (Magnoflorine) is an aporphine alkaloid found in Acoruscalamus, with anti-fungal activity, reduces the formation of C. albicans’ biofilm[1]. Anti-antidiabeticand anti-oxidative activity[2].

  • CAS Number: 2141-09-5
  • MF: C20H24NO4+
  • MW: 342.408
  • Catalog: Fungal
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: 252ºC
  • Flash Point: N/A