An antifungal agent is a drug that selectively eliminates fungal pathogens from a host with minimal toxicity to the host. Classes: 1. Polyene Antifungal Drugs: Amphotericin, nystatin, and pimaricin interact with sterols in the cell membrane (ergosterol in fungi, cholesterol in humans) to form channels through which small molecules leak from the inside of the fungal cell to the outside. 2. Azole Antifungal Drugs: Fluconazole, itraconazole, and ketoconazole inhibit cytochrome P450-dependent enzymes (particularly C14-demethylase) involved in the biosynthesis of ergosterol, which is required for fungal cell membrane structure and function. 3. Allylamine and Morpholine Antifungal Drugs: lylamines (naftifine, terbinafine) inhibit ergosterol biosynthesis at the level of squalene epoxidase. The morpholine drug, amorolfine, inhibits the same pathway at a later step. 4. Antimetabolite Antifungal Drugs: 5-Fluorocytosine acts as an inhibitor of both DNA and RNA synthesis via the intracytoplasmic conversion of 5-fluorocytosine to 5-fluorouracil.


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Mancozeb

Mancozeb is an ethylene-bis-dithiocarbamate fungicide[1].

  • CAS Number: 8018-01-7
  • MF: C8H12Mn2N4S8Zn22-
  • MW: 661.36
  • Catalog: Fungal
  • Density: 1.92 g/cm3
  • Boiling Point: 308.2ºC at 760 mmHg
  • Melting Point: 192-194°C
  • Flash Point: 138 °C

Triphala

Triphala, an Ayurvedic polyherbal formulation comprising of equiproportional fruit parts of Terminalia chebula, Terminalia bellerica, and Phyllanthus emblica[1]. Triphala inhibits NF-κB activation. Triphala exerts antifungal action[2]. Anti-adipogenic, anti-inflammatory, and anti-neoplastic activities.

  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Lithium benzoate

Benzoic acid (lithium) is an aromatic alcohol found in many plants and is a common additive in food, beverages, cosmetics and other products. Benzoic acid (lithium) inhibits bacteria and fungi and acts as a preservative[1].

  • CAS Number: 553-54-8
  • MF: C7H5LiO2
  • MW: 128.05
  • Catalog: Bacterial
  • Density: 1.19g/cm3
  • Boiling Point: 249.3ºC at 760 mmHg
  • Melting Point: >300 °C(lit.)
  • Flash Point: 111.4ºC

Monomyristin

1-Monomyristin, extracted from Serenoa repens, inhibits the hydrolysis of 2-oleoylglycerol (IC50=32 μM) and fatty acid amide hydrolase (FAAH) activity (IC50=18 μM). 1-Monomyristin shows antibacterial activity against Staphylococcus aureus and Aggregatibacter actinomycetemcomitans and also antifungal activity against Candida albicans[1][2][3].

  • CAS Number: 589-68-4
  • MF: C17H34O4
  • MW: 302.449
  • Catalog: Bacterial
  • Density: 1.0±0.1 g/cm3
  • Boiling Point: 424.8±25.0 °C at 760 mmHg
  • Melting Point: 68-70ºC
  • Flash Point: 141.3±16.7 °C

Micafungin Sodium

Micafungin sodium (FK 463) is an antifungal agent which inhibits 1, 3-beta-D-glucan synthesis.

  • CAS Number: 208538-73-2
  • MF: C56H70N9NaO23S
  • MW: 1292.256
  • Catalog: Fungal
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Harzianum A

Harzianum A is a trichothecene that isolated from the soil-borne fungus Trichoderma harzianum. Harzianum A shows no cytotoxicity against baby hamster kidney cells, no activity against Gram-negative and Gram-positive bacteria, but modest antifungal activity at 100 μg/mL[1].

  • CAS Number: 156250-74-7
  • MF: C23H28O6
  • MW: 400.46500
  • Catalog: Fungal
  • Density: 1.26g/cm3
  • Boiling Point: 556.9ºC at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 190.1ºC

Me1111

ME1111 is an antifungal agent that is active against dermatophytes. ME1111 is an inhibitor of the succinate dehydrogenase of Trichophyton species. ME1111 has an excellent ability to penetrate human nails and is used for onychomycosis research[1][2].

  • CAS Number: 1391758-52-3
  • MF: C12H14N2O
  • MW: 202.25
  • Catalog: Fungal
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Antifungal agent 24

Antifungal agent 24 (Compound 6) is an antifungal agent against Candida albicans with a MIC value of 0.03 μg/mL[1].

  • CAS Number: 2566522-60-7
  • MF: C24H18F2N4O
  • MW: 416.42
  • Catalog: Fungal
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Isoliquiritoside

Isoliquiritin, isolated from Licorice Root, inhibits angiogenesis and tube formation. Isoliquiritin also exhibits antidepressant-like effects and antifungal activity[1][2][3].

  • CAS Number: 5041-81-6
  • MF: C21H22O9
  • MW: 418.394
  • Catalog: Fungal
  • Density: 1.5±0.1 g/cm3
  • Boiling Point: 743.5±60.0 °C at 760 mmHg
  • Melting Point: 185-186ºC
  • Flash Point: 263.3±26.4 °C

Faltan-d4

Faltan-d4 is the deuterium labeled Faltan[1]. Faltan is a dicarboximide fungicide, widely used on vines and several vegetable crops, and is also cytotoxic effect on human bronchial epithelial cells[2].

  • CAS Number: 1327204-12-5
  • MF: C9D4Cl3NO2S
  • MW: 300.582
  • Catalog: Fungal
  • Density: 1.7±0.1 g/cm3
  • Boiling Point: 333.8±52.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 155.7±30.7 °C

Tetrahydrojatrorrhizine

Corypalmine is an alkaloid from Corydalis chaerophylla. Corypalmine is an antifungal.

  • CAS Number: 27313-86-6
  • MF: C20H23NO4
  • MW: 341.40100
  • Catalog: Fungal
  • Density: 1.29g/cm3
  • Boiling Point: 501.2ºC at 760mmHg
  • Melting Point: N/A
  • Flash Point: 256.9ºC

Antifungal agent 31

Antifungal agent 31 (compound 12) is a potent and orally active triazole antifungal agents with a pyrrolotriazinone scaffold. Antifungal agent 31 shows antifungal activity against Candida spp. and filamentous fungi. Antifungal agent 31 significantly reduced mortality rates and kidney fungal burden in two murine models of lethal systemic infections[1].

  • CAS Number: 2077083-94-2
  • MF: C25H22F2N6O3
  • MW: 492.48
  • Catalog: Fungal
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

JUSTICIDIN B

Justicidin B is a potent anticancer lignan and proapoptotic agent. Justicidin B is also a bone resorption inhibitor, and has strong antiviral, fungicidal, antiprotozoal effects. Justicidin B significantly inhibits platelet aggregation[1][2][3].

  • CAS Number: 17951-19-8
  • MF: C21H16O6
  • MW: 364.34800
  • Catalog: Fungal
  • Density: 1.376g/cm3
  • Boiling Point: 601.9ºC at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 266ºC

(+)-Piresil diacetate

(+)-Pinoresinol diacetate is an antifungal agent that can be isolated from Sambucus williamsii[1].

  • CAS Number: 32971-25-8
  • MF: C24H26O8
  • MW: 442.458
  • Catalog: Fungal
  • Density: 1.2±0.1 g/cm3
  • Boiling Point: 539.9±50.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 232.4±30.2 °C

Pseudolaric Acid A

Pseudolaric Acid A is a diterpene acid isolated from Pseudolarix kaempferi, has antifungal, cytotoxic and antifertile activities[1][2][3].

  • CAS Number: 82508-32-5
  • MF: C22H28O6
  • MW: 388.454
  • Catalog: Fungal
  • Density: 1.23
  • Boiling Point: 571.5±50.0 °C at 760 mmHg
  • Melting Point: 206-207 ºC
  • Flash Point: 196.6±23.6 °C

TMV-IN-5

TMV-IN-5 (compound 1a) is an anti-plant virus/fungal agent. TMV-IN-5 inhibits viral assembly by binding to tobacco mosaic virus (TMV) CP. TMV-IN-5 can be used in the development of pesticides[1].

  • CAS Number: 1207318-92-0
  • MF: C22H23N3S
  • MW: 361.50
  • Catalog: Fungal
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Fenpropidin

Fenpropidin is a sterol biosynthesis inhibitor fungicide[1].

  • CAS Number: 67306-00-7
  • MF: C19H31N
  • MW: 273.45600
  • Catalog: Fungal
  • Density: 0.924 g/cm3
  • Boiling Point: 368.9ºC at 760 mmHg
  • Melting Point: 25°C
  • Flash Point: 159.3ºC

Oligomycin

Oligomycins are macrolides created by Streptomyces species that can be toxic to other organisms through their ability to inhibit mitochondrial membrane-bound ATP synthases. The mitochondrial F1FO ATP synthase can switch to an ATP hydrolase during ischemia, so that, under these conditions, inhibition by oligomycins will reduce ATP depletion rather than block ATP synthesis.

  • CAS Number: 1404-19-9
  • MF: C135H220O33
  • MW: 2371.171
  • Catalog: Fungal
  • Density: 1.14 g/cm3
  • Boiling Point: 886.3ºC at 760 mmHg
  • Melting Point: 84-100ºC
  • Flash Point: 252ºC

Tolnaftate-d7

Tolnaftate D7 (NP-27 D7) is the deuterium labeled Tolnaftate. Tolnaftate (NP-27) is a synthetic thiocarbamate used as an anti-fungal agent[1][2].

  • CAS Number: 1329835-64-4
  • MF: C19H10D7NOS
  • MW: 314.453
  • Catalog: Fungal
  • Density: 1.2±0.1 g/cm3
  • Boiling Point: 453.4±38.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 228.0±26.8 °C

Tolytoxin

Tolytoxin, a bioactive metabolite from cyanobacteria, is a potent antifungal antibiotic, exhibiting MICs of 0.25-8 nmol. Tolytoxin is a cyanobacterial macrolide that targets actin by inhibition of its polymerization. Tolytoxin has cytotoxic effects in cancer cells[1].

  • CAS Number: 127999-44-4
  • MF: C46H75NO13
  • MW: 850.09
  • Catalog: Fungal
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Agoniadin

Plumieride is an antifungal agent. Plumieride has strong fungitoxicity against some dermatophytes. Plumieride has little cytotoxic activity against the P388 leukaemia cell line with an IC50 of 85 μg/mL[1].

  • CAS Number: 511-89-7
  • MF: C21H26O12
  • MW: 470.42
  • Catalog: Fungal
  • Density: 1.6±0.1 g/cm3
  • Boiling Point: 771.4±60.0 °C at 760 mmHg
  • Melting Point: 156-158°; mp 224-225°
  • Flash Point: 269.2±26.4 °C

Fmoc-Gly-OH-1-13C

Fmoc-Gly-OH-1-13C is a 13C-labeled Carbendazim. Carbendazim is a potent and orally active broad-spectrum benzimidazole fungicide and can be acts as a pesticide for fungal diseases research, such as Seproria, Fusarium and Sclerotina[1][3]. Carbendazim is a

  • CAS Number: 197965-68-7
  • MF: C1613CH15NO4
  • MW: 298.30
  • Catalog: Fungal
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Sakuranetin

Sakuranetin is a rice flavonoid phytoalexin, shows strong antifungal activity[1]. Sakuranetin has anti-inflammatory and antioxidative activities. Sakuranetin ameliorates LPS-induced acute lung injury[2].

  • CAS Number: 2957-21-3
  • MF: C16H14O5
  • MW: 286.28
  • Catalog: Fungal
  • Density: 1.4±0.1 g/cm3
  • Boiling Point: 555.9±50.0 °C at 760 mmHg
  • Melting Point: 153-154ºC
  • Flash Point: 212.4±23.6 °C

Magnoflorine

(+)-Magnoflorine (Magnoflorine) is an aporphine alkaloid found in Acoruscalamus, with anti-fungal activity, reduces the formation of C. albicans’ biofilm[1]. Anti-antidiabeticand anti-oxidative activity[2].

  • CAS Number: 2141-09-5
  • MF: C20H24NO4+
  • MW: 342.408
  • Catalog: Fungal
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: 252ºC
  • Flash Point: N/A

(E)-β-Farnesene

(E)-β-Farnesene (trans-β-Farnesene) is a volatile sesquiterpene hydrocarbon which can be found in Phlomis aurea Decne essential oil. (E)-β-Farnesene can be used as a feeding stimulant for the sand fly Lutzomyia longipalpis[1][2].

  • CAS Number: 18794-84-8
  • MF: C15H24
  • MW: 204.35100
  • Catalog: Fungal
  • Density: 0.807 g/cm3
  • Boiling Point: 272.5ºC at 760 mmHg
  • Melting Point: < 25ºC
  • Flash Point: 230°F(110ºC)

Meridinol

Meridinol ((-)-Meridinol) shows antimicrobial activity against a wide range of gram-positive and gram-negative bacteria and fungi.

  • CAS Number: 120051-54-9
  • MF: C20H18O7
  • MW: 370.353
  • Catalog: Bacterial
  • Density: 1.5±0.1 g/cm3
  • Boiling Point: 565.8±45.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 205.1±22.2 °C

Methyl 7-formylcyclopenta[c]pyran-4-carboxylate

Cerbinal is a natural compound isolated from Gardenia jasminoides Ellis. Cerbinal has antifungal activity[1].

  • CAS Number: 65597-42-4
  • MF: C11H8O4
  • MW: 204.179
  • Catalog: Fungal
  • Density: 1.3±0.1 g/cm3
  • Boiling Point: 433.4±40.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 198.8±27.4 °C

Thiophanate-methyl-d6

Thiophanate-methyl-d6 is the deuterium labeled Thiophanate-methyl. Thiophanate-Methyl is a systematic fungicide[1][2].

  • CAS Number: 1398065-77-4
  • MF: C12H8D6N4O4S2
  • MW: 348.43
  • Catalog: Fungal
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

5-Aminouridine

5-Aminouridine can modify nucleobases and can be incorporated into the target DNA. 5-Aminouridine exhibits a wide range of biological activity and it inhibits the growth of tumors, fungi and viruses[1][2][3].

  • CAS Number: 2149-76-0
  • MF: C9H13N3O6
  • MW: 259.21600
  • Catalog: Fungal
  • Density: 1.712g/cm3
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Rimocidin

Rimocidin, a polyene macrolide, is an antifungal compound. Rimocidin shows broad‐spectrum antifungal activity against multiple plant‐pathogenic fungi[1][2].

  • CAS Number: 1393-12-0
  • MF: C39H61NO14
  • MW: 767.90000
  • Catalog: Fungal
  • Density: 1.34g/cm3
  • Boiling Point: 1039.5ºC at 760mmHg
  • Melting Point: N/A
  • Flash Point: 582.5ºC